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IDPMIDSEQUENCENAME LENGTHACTIVITY
105318617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=14.7 µg/ml
105418617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=11.3 µg/ml
105518617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=8.2 µg/ml
105618617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=17 µg/ml
105718617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=10.5 µg/ml
105818617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=20.2 µg/ml
114112005420KWKLFKKIPKFLHSAKKFCA-MA-P18IC50=20 µM
114212005420KWKFKKIPKFLHLAKKFP1817IC50=4 µM
114312005420KWKLFKKILKFLHLAKKF[L9]-P1818IC50=9 µM
114412005420KWKLFKKISKFLHLAKKF[S9]-P1818IC50=7 µM
114512005420WKLFKKIPKFLHLAKKFN-117IC50=12 µM
114612005420FKLFKKIPKFLHLAKKFN-217IC50=11 µM
114712005420KWFKKIPKFLHLAKKFN-316IC50=17 µM
114812005420WFKKIPKFLHLAKKFN-415IC50=23 µM
114912005420WKKIPKFLHLAKKFN-514IC50=100.0 <µM
115012005420KWFKKIPKFLHLLKKFN-3L16IC50=4 µM
115112005420WFKKIPKFLHLLKKFN-4L15IC50=6 µM
115212005420WKKIPKFLHLLKKFN-5L14IC50=14 µM
115312005420KWKLFKKIPFLHLAKKFC-117IC50=32 µM
115412005420KWKLFKKIPKFLHLAKKC-217IC50=26 µM
115512005420KWKLFKKIPLHLAKKFC-316IC50=74 µM
115612005420KWKLFKKIPKFLHLAKC-416IC50=31 µM
115712005420KWKLFKKIPHLAKKFC-515IC50=81 µM
115812005420KWKLFKKIPKFLHLAC-615IC50=21 µM
115912005420KWKLFKKIPLAKKFC-714IC50=100.0 <µM
116012005420KWKLFKKIPKFLHLC-814IC50=54 µM
116112005420KWKLFKKIPLKKFC-913IC50=100.0 <µM
116212005420KWKLFKKIPKFLHC-1013IC50=100.0 <µM
116312005420KWKLFKKIPKFLHSAKKFCA-MA-P18IC50=25 µM
116412005420KWKFKKIPKFLHLAKKFP1817IC50=3.5 µM
116512005420KWKLFKKILKFLHLAKKF[L9]-P1818IC50=3 µM
116612005420KWKLFKKISKFLHLAKKF[S9]-P1818IC50=3 µM
116712005420WKLFKKIPKFLHLAKKFN-117IC50=6 µM
116812005420FKLFKKIPKFLHLAKKFN-217IC50=7 µM
116912005420KWFKKIPKFLHLAKKFN-316IC50=11 µM
117012005420WFKKIPKFLHLAKKFN-415IC50=24 µM
117112005420WKKIPKFLHLAKKFN-514IC50=100.0 <µM
117212005420KWFKKIPKFLHLLKKFN-3L16IC50=4.2 µM
117312005420WFKKIPKFLHLLKKFN-4L15IC50=3 µM
117412005420WKKIPKFLHLLKKFN-5L14IC50=10 µM
117512005420KWKLFKKIPFLHLAKKFC-117IC50=31 µM
117612005420KWKLFKKIPKFLHLAKKC-217IC50=23 µM
117712005420KWKLFKKIPLHLAKKFC-316IC50=62 µM
117812005420KWKLFKKIPKFLHLAKC-416IC50=25 µM
117912005420KWKLFKKIPHLAKKFC-515IC50=67 µM
118012005420KWKLFKKIPKFLHLAC-615IC50=27 µM
118112005420KWKLFKKIPLAKKFC-714IC50=100.0 <µM
118212005420KWKLFKKIPKFLHLC-814IC50=30 µM
118312005420KWKLFKKIPLKKFC-913IC50=100.0 <µM
118412005420KWKLFKKIPKFLHC-1013IC50=100.0 <µM
118510675500KWKLFKKIGIGKFLHSAKKFCA-MA20IC50=65 µM
118610675500KWKLFKKIKFLHSAKKFCA-MA117IC50=85.3 µM
118710675500KWKLFKKIPKFLHSAKKFCA-MA218IC50=35.1 µM
118810675500KWKLFKKIGPGKFLHSAKKFCA-MA320IC50=>100 µM
119310675500KWKLFKKIGIGKFLHSAKKFCA-MA20IC50=30 µM
119410675500KWKLFKKIKFLHSAKKFCA-MA117IC50=65 µM
119510675500KWKLFKKIPKFLHSAKKFCA-MA218IC50=20 µM
119610675500KWKLFKKIGPGKFLHSAKKFCA-MA320IC50=75 µM
12317849420KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKALCecropin B35IC50=15.5 µM
12357849420SWLSKTAKKLENSAKKRISEGIAIAIQGGPRCecropin P131IC50=93 µM
12397849420MPRWRLFRRIDRVGKQIKQGILRAGPAIALVGDARAVGShiva-138IC50=28.7 µM
12437849420KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKALCecropin B35IC50=4.4 µM
125310951191GLFDIIKKIAESFAurein1.213LC50=10-100 µM
126210951191GLFDIVKKVVGAFGSLAurein2.516LC50=10-100 µM
127110951191GLFDIAKKVIGVIGSLAurein2.616LC50=10-100 µM
128010951191GLFDIVKKIAGHIAGSIAurein 3.117LC50 = 10 µM
128910951191GLFDIVKKIAGHIASSIAurein 3.217LC50 = 10 µM
129810951191GLFDIVKKIAGHIVSSIAurein 3.317LC50=10-100 µM
135218425992FKCRRWQWRMKKLGAPSITCVRpep122IC50=77 µM
135318425992RKAFRWAWRMLKKAAPSITCVRmPep122IC50=8 µM
13541708887, 2285300GIGKFLHAAKKFAKAFVAEIMNSMagainin B23IC50=17 µg/ml
13551708887, 2285300GIGKFLHSAKKFAKAFVAEIMNSMagainin G23IC50=19 µg/ml
13561708887, 2285300AIGKFLHSAKKFGKAFVGEIMNSMagainin A23IC50=16 µg/ml
13571708887, 2285300ALSKALSKALSKALSKALSKALSKZ4424IC50=97 µg/ml
13581708887, 2285300ALSKALSKALSKALSKALSKALSKZ2424IC50=123 µg/ml
13591708887, 2285300GIGKFLHSAKKFGKAFVGEIMNSMagainin 223IC50 >150 µg/ml
13601708887, 2285300GIGKFLHAAKKFAKAFVAEIMNSMagainin B23IC50=12 µg/ml
13611708887, 2285300GIGKFLHSAKKFAKAFVAEIMNSMagainin G23IC50=16 µg/ml
13621708887, 2285300AIGKFLHSAKKFGKAFVGEIMNSMagainin A23IC50=18 µg/ml
13631708887, 2285300ALSKALSKALSKALSKALSKALSKZ4424IC50=60 µg/ml
13641708887, 2285300ALSKALSKALSKALSKALSKALSKZ2424IC50=83 µg/ml
13651708887, 2285300GIGKFLHSAKKFGKAFVGEIMNSMagainin 223IC50 >150 µg/ml
13661708887, 2285300GIGKFLHAAKKFAKAFVAEIMNSMagainin B23IC50=27 µg/ml
13671708887, 2285300GIGKFLHSAKKFAKAFVAEIMNSMagainin G23IC50=29 µg/ml
13681708887, 2285300AIGKFLHSAKKFGKAFVGEIMNSMagainin A23IC50=23 µg/ml
13691708887, 2285300ALSKALSKALSKALSKALSKALSKZ4424IC50=107 µg/ml
13701708887, 2285300ALSKALSKALSKALSKALSKALSKZ2424IC50=109 µg/ml
13711708887, 2285300GIGKFLHSAKKFGKAFVGEIMNSMagainin 223IC50 >150 µg/ml
13721708887, 2285300GIGKFLHAAKKFAKAFVAEIMNSMagainin B23IC50=28 µg/ml
13731708887, 2285300GIGKFLHSAKKFAKAFVAEIMNSMagainin G23IC50=38 µg/ml
13741708887, 2285300AIGKFLHSAKKFGKAFVGEIMNSMagainin A23IC50=30 µg/ml
13751708887, 2285300ALSKALSKALSKALSKALSKALSKZ4424IC50=115 µg/ml
13761708887, 2285300ALSKALSKALSKALSKALSKALSKZ2424IC50=143 µg/ml
13771708887, 2285300GIGKFLHSAKKFGKAFVGEIMNSMagainin 223IC50 >150 µg/ml
13781708887, 2285300GIGKFLHAAKKFAKAFVAEIMNSMagainin B23IC50=30 µg/ml
13791708887, 2285300GIGKFLHSAKKFAKAFVAEIMNSMagainin G23IC50=33 µg/ml
13801708887, 2285300AIGKFLHSAKKFGKAFVGEIMNSMagainin A23IC50=34 µg/ml
13811708887, 2285300ALSKALSKALSKALSKALSKALSKZ4424IC50=80 µg/ml
13821708887, 2285300ALSKALSKALSKALSKALSKALSKZ2424IC50=102 µg/ml
13831708887, 2285300GIGKFLHSAKKFGKAFVGEIMNSMagainin 223IC50 >150 µg/ml
13841708887, 2285300GIGKFLHAAKKFAKAFVAEIMNSMagainin B23IC50=23 µg/ml
13851708887, 2285300GIGKFLHSAKKFAKAFVAEIMNSMagainin G23IC50=25 µg/ml
13861708887, 2285300AIGKFLHSAKKFGKAFVGEIMNSMagainin A23IC50=20 µg/ml
13871708887, 2285300ALSKALSKALSKALSKALSKALSKZ4424IC50=64 µg/ml
13881708887, 2285300ALSKALSKALSKALSKALSKALSKZ2424IC50=72 µg/ml
13891708887, 2285300GIGKFLHSAKKFGKAFVGEIMNSMagainin 223IC50 >150 µg/ml
13901708887, 2285300GIGKFLHAAKKFAKAFVAEIMNSMagainin B23IC50=32 µg/ml
13911708887, 2285300GIGKFLHSAKKFAKAFVAEIMNSMagainin G23IC50=37 µg/ml
13921708887, 2285300AIGKFLHSAKKFGKAFVGEIMNSMagainin A23IC50=40 µg/ml
13931708887, 2285300ALSKALSKALSKALSKALSKALSKZ4424IC50=98 µg/ml
13941708887, 2285300ALSKALSKALSKALSKALSKALSKZ2424IC50=112 µg/ml
13951708887, 2285300GIGKFLHSAKKFGKAFVGEIMNSMagainin 223IC50 >150 µg/ml
13961708887, 2285300GIGKFLHAAKKFAKAFVAEIMNSMagainin B23IC50=32 µg/ml
13971708887, 2285300GIGKFLHSAKKFAKAFVAEIMNSMagainin G23IC50=39 µg/ml
13981708887, 2285300AIGKFLHSAKKFGKAFVGEIMNSMagainin A23IC50=45 µg/ml
13991708887, 2285300ALSKALSKALSKALSKALSKALSKZ4424Not Available
14001708887, 2285300ALSKALSKALSKALSKALSKALSKZ2424Not Available
14011708887, 2285300GIGKFLHSAKKFGKAFVGEIMNSMagainin 223IC50 >200 µg/ml
14208573171, 21403917TRSSRAGLQFPVGRVHRLLRKBuforin2215% Cytotoxicity at 0.5 µg/ml
142110455241, 21403917GLFDVIKKVASVIGGLCitropin1.11660% Cytotoxicity at 0.5 µg/ml
142210504394, 21403917GLFDVIKKVASVIGGLCitropin1.11660% Cytotoxicity at 0.5 µg/ml
142316512752, 21403917AKRHHGYKRKFHDemegen P-1131215% Cytotoxicity at 0.5 µg/ml
142414508884, 21403917ILRWPWWPWRRKOmigaNAn MBI-2261227% Cytotoxicity at 0.5 µg/ml
14257768152, 21403917GIGKFLKKAKKFGKAFVKILKKPexigaNAn MSI-782275% Cytotoxicity at 0.5 µg/ml
14268335113, 21403917RGGRLCYCRRRFCVCVGRProtegrin 11861% Cytotoxicity at 0.5 µg/ml
14279022710FLPLIGRVLSGILTemporin A1315% Cytotoxicity at 0.5 µg/ml
143016269280KILRGVCKKIMRTFLRRISKDILTGKKNK-227LD50=30 µM
143116269280KILRGVCKKIMRTFLRRISKDILTGKKNK-227LD50=1-4 µM
164911835991GIGTKILGGVKTALKGALKELASTYANmaximin127IC50=15.3 µg/ml
165011835991GIGGKILSGLKTALKGAAKELASTYLHmaximin327IC50=11.4 µg/ml
165111835991GIGVLLSAGKAALKGLAKVLAEKYANmaximin426IC50=24.2 µg/ml
165211835991SIGAKILGGVKTFFKGALKELASTYLQmaximin527IC50=34.4 µg/ml
165311835991GIGTKILGGVKTALKGALKELASTYANmaximin127IC50=24.3 µg/ml
165411835991GIGGKILSGLKTALKGAAKELASTYLHmaximin327IC50 =25.2 µg/ml
165511835991GIGVLLSAGKAALKGLAKVLAEKYANmaximin426IC50 =53.4 µg/ml
165611835991SIGAKILGGVKTFFKGALKELASTYLQmaximin527IC50 >50 µg/ml
282223000474RRRRRNWMWC9R10IC50=93 µM
282323000474RRRRRWCMNW9S1R10IC50=38 µM
282423000474RRRRRNWMWC9R10IC50=39 µM
282523000474RRRRRWCMNW9S1R10IC50=43 µM
282623000474RRRRRNWMWC9R10IC50=37 µM
282723000474RRRRRWCMNW9S1R10IC50=43 µM
282823000474RRRRRNWMWC9R10IC50=36 µM
282923000474RRRRRWCMNW9S1R10IC50=45 µM
283023000474RRRRRNWMWC9R10IC50=25 µM
283123000474RRRRRWCMNW9S1R10IC50=36 µM
283223000474RRRRRNWMWC9R10IC50=47 µM
283323000474RRRRRWCMNW9S1R10IC50=26 µM
283423000474RRRRRNWMWC9R10IC50=12 µM
283523000474RRRRRWCMNW9S1R10IC50=17 µM
284224246647GIIKKIIKKIShort α-helical peptides10100% Cytotoxicity at 5 µM Approx
284324246647GIIKKIIKKIIKKIShort α-helical peptides1490% Cytotoxicity at 5 µM Approx
284424246647GIIKKIIKKIIKKIIKKIShort α-helical peptides1870% Cytotoxicity at 5 µM Approx
285023028527GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAVAdenoregulin33GI50 =2.57±0.75 µM
307216004618MRKEFHNVLSSGQLLADKRPARDYNRKPep2727Not Available
307316004618MWKWFHNVLSSWQLLADKRPARDYNRKPep27anal127IC50= 50 µM
307416004618MWKWFHNVLSWWWLLADKRPARDYNRKPep27anal227IC50= 29 µM
307516004618MRKWFHNVLSSGQLLADKWPAWDYNRKPep27anal327IC50= 67 µM
307616004618MWKEFHNVLSSGQLLADKRWARWYNRWPep27anal427IC50= 50 µM
307716004618MWKWFHNVLSSGQLLADKWWAWWYNWWPep27anal527IC50= >70 µM
307816004618MRKEFHNVLSSGQLLADKRPARDYNRKPep2727IC50= >70 µM
307916004618MWKWFHNVLSSWQLLADKRPARDYNRKPep27anal127IC50= 53 µM
308016004618MWKWFHNVLSWWWLLADKRPARDYNRKPep27anal227IC50= 20 µM
308116004618MRKWFHNVLSSGQLLADKWPAWDYNRKPep27anal327IC50= 52 µM
308216004618MWKEFHNVLSSGQLLADKRWARWYNRWPep27anal427IC50=51 µM
308316004618MWKWFHNVLSSGQLLADKWWAWWYNWWPep27anal527IC50= >70 µM
308416004618MRKEFHNVLSSGQLLADKRPARDYNRKPep2727IC50=>70 µM
308516004618MWKWFHNVLSSWQLLADKRPARDYNRKPep27anal127IC50= 47 µM
308616004618MWKWFHNVLSWWWLLADKRPARDYNRKPep27anal227IC50= 23 µM
308716004618MRKWFHNVLSSGQLLADKWPAWDYNRKPep27anal327IC50= 50 µM
308816004618MWKEFHNVLSSGQLLADKRWARWYNRWPep27anal427IC50= 46 µM
308916004618MWKWFHNVLSSGQLLADKWWAWWYNWWPep27anal527IC50=>70 µM
310422783018PDEDAINNALNKVCSTGRRQRSICKQLLKKN29N30100% cell viability at 5 µM
310522783018PDEDAINNALNKVCSTGRRQRSICKQLLKKN29N30<40% cell viability at 50 µM
311022783018PDEDAINDALNKVCSTGRRQRSICKQLLKKN29D30100% cell viability at 5 µM
311122783018PDEDAINDALNKVCSTGRRQRSICKQLLKKN29D30<60% cell viability at 50 µM
315723301519WRWRWRWRWCyclic [W(RW)4 ]-Dox962-73% inhibition of cell proliferation at 1 µM
316123301519RWRWRWRWlinear (RW)4-Dox846-69% antiproliferative activity at 1 µM
318017559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 54010.4 % inhibition of cell proliferation at 1 nM
318117559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 54018.7 % inhibition of cell proliferation at 10 nM
318217559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 54034.7 % inhibition of cell proliferation at 100 nM
318317559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 54054.3 % inhibition of cell proliferation at 1 µM
318417559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 54094.5 % inhibition of cell proliferation at 10 µM
318817559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 540ED50 =0.29 µM
325622783018PDEDAINNALNKVCSTGRRQRSICKQLLKKN29N30100% cell viability at 5 µM
325722783018PDEDAINNALNKVCSTGRRQRSICKQLLKKN29N30<40% cell viability at 50 µM
326222783018PDEDAINDALNKVCSTGRRQRSICKQLLKKN29D30100% cell viability at 5 µM
326322783018PDEDAINDALNKVCSTGRRQRSICKQLLKKN29D30<60% cell viability at 50 µM
328319527490, 23533710FKCRRWQWRMKKLfcinB12IC50 = 55 µM
328619527490, 23533710FKCRRWQWRMKKLfcinB12IC50 = 13 µM
328719527490, 23533710FKCRRWQWRMKKLfcinB12IC50 = 10 µM
334522820149Structure GivenBAA-1Not AvailableIC50 = 8.1 µg/ml
334622820149Structure GivenBAA-2Not AvailableIC50 = 3.8 µg/ml
3352NoneKWKLFKKIGIGKFLHSAKKFCA-MA20100% survival rate at 10 µM
3353NoneKWKLFKKIGIGKFLHSAKKFCA-MA200% survival rate at 100 µM
3358NoneKWKKLLKKPPPLLKKLLKKLSynthetic peptide20~60% survival rate at 10 µM
3359NoneKWKKLLKKPPPLLKKLLKKLSynthetic peptide200% survival rate at 100 µM
354522100226VNWKKILGKIIKVVKLL-III15IC50 = 5±3 µM
354622100226VNWKKILAKIIKVVKLL-III/115IC50 = 3±1 µM
354722100226NVWKKILGKIIKVVKLL-III/215IC50 = 7±2 µM
354822100226VNWKKILKKIIKVVKLL-III/315Not tested
354922100226VNWKKILGKIKKVVKLL-III/415IC50 = 18 µM
355022100226VNWKKILPKIIKVVKLL-III/615IC50 = 6±3 µM
355122100226VNWKKILGKIIKVVKLL-III/815IC50 = 9 µM
355222100226VNWKKILGKIIKVVKLL-III/915Not tested
355322100226KNWKKILGKIIKVVKLL-III/1015IC50 = 9 µM
355422100226VNWKKIILGKIIKVVKLL-III/1115IC50 = 4±1 µM
355522100226vnwkkilgkiikvvkLL-III/1215IC50 = 5±2 µM
355622100226VNFKKLLGKLLKVVKLL-III/1515IC50 = 9±3 µM
355722100226VN-Nal-KKLLGKLLKVVKLL-III/1615Not tested
355822100226VNWRRILGRIIRVVRLL-III/1715Not tested
355922100226KNWKKILKKIIKVVKLL-III/1815IC50 = 7±2 µM
356022100226VNWKK-Aib-LGK-Aib-IK-Aib-VKLL-III/1915IC50 = 8±2 µM
356122100226KNWKK-Aib-LKK-Aib-IK-Aib-VKLL-III/2215IC50 = 25±4 µM
356222100226VNWKKLLGKLLKVVKLL-III/2315IC50 = 6 µM
356322100226VNWOOILGOIIOVVOLL-III/2415IC50 = 5±2 µM
356422100226vnwkkllgkllkvvkLL-III/2515IC50 = 4 µM
356522100226VYWKKILGKIIKVVKLL-III/2615IC50 = 6 µM
356622100226VNWKKVLGKVVKVVKLL-III/2715IC50 = 18 µM
356722100226NKWKKILGKIIKVVKLL-III/3415IC50 = 5±3 µM
356822100226VNWKKILAKIIKVVKLL-III/3615Not tested
356922100226VNWKKILGKIIKVVKLL-III/3715IC50= 4±1 µM
361822100226GFGMALKLLKKVLMAC113IC50 = 12±6 µM
361922100226GTGLPMSERRKIMLMMRMAC217IC50 = 32 µM
362022100226gfgmalkllkkvlMAC1/113IC50 = 11 µM
362122100226AFGMALKLLKKVLMAC1/213IC50 = 17 µM
362222100226LFGMALKLLKKVLMAC1/313IC50 = 22 µM
362322100226GFGMALKLLKKVLMAC1/413IC50 = 29 µM
362422100226GFGMALKLLKKVLMAC1/613IC50 = 15 µM
362522100226GFKMALKLLKKVLMAC1/913IC50 = 14±4 µM
362622100226GFKMALKLLKKVLMAC1/1013IC50 = 16 µM
362722100226GFGMALKLLKKVLMAC1/1613IC50 = 70 µM
362822100226GFGMALKLLKKVLMAC1/1913IC50 = 43±11 µM
362922100226GFGMALOLLOOVLMAC1/2013IC50 = 25±3 µM
363022100226GFGMALRLLRRVLMAC1/2113IC50 = 22±4 µM
363122100226GFGMALKL-(AC6C)-KKVLMAC1/2413IC50 = 11 µM
363222100226GFGMALK-(AC6C)-LKKVLMAC1/2513IC50 = 12±2 µM
363322100226GFGMA-(AC6C)-KLLKKVLMAC1/2613IC50 = 9±2 µM
369022100226GMWSKILGHLIRHAL-112IC50 = 49±9 µM
369122100226gmwskilghlirHAL-1/2212Not tested
369222100226GMWSKILGHLIKHAL-1/612Not tested
369322100226GMWSKILGHLKRHAL-1/412Not tested
369422100226GMWSKILGKLIRHAL-1/912IC50 = 30±10 µM
369522100226GMWSKILKHLIRHAL-1/1812Not tested
369622100226GMWKKILGHLIRHAL-1/512IC50 > 40 µM
369722100226GKWSKILGHLIRHAL-1/1212IC50 > 40 µM
369822100226KMWSKILGHLIRHAL-1/1712Not tested
369922100226GMWKKILGKLIRHAL-1/1012Not tested
370022100226GKWSKILGKLIRHAL-1/2012IC50 > 40 µM
370122100226GKWKKILGHLIRHAL-1/1912Not tested
370222100226GKWKKILGKLIRHAL-1/2112Not tested
370322100226GMWSKILGHLIRHAL-1/2912Not tested
370422100226GMWSKLLGHLLRHAL-1/1512IC50 > 40 µM
370522100226GKWMSLLKHILKHAL-212IC50 = 34 µM
370622100226gkwmsllkhilkHAL-2/2212Not tested
370722100226GKWMSLLKKILKHAL-2/412Not tested
370822100226GKWMKLLKHILKHAL-2/212IC50 > 40 µM
370922100226GKWKSLLKHILKHAL-2/112IC50 > 40 µM
371022100226GKWMSLLKHILKHAL-2/812Not tested
371122100226GKWMSLLKHIWKHAL-2/1812Not tested
371222100226GKWMSLLKHWLKHAL-2/1912Not tested
371322100226GKWMSLWKHILKHAL-2/2012Not tested
371422100226GKFMSLLKHILKHAL-2/2412Not tested
371522100226GKWMSFLKHILKHAL-2/612Not tested
371622100226GKWMTLLKHILKHAL-2/1312Not tested
371722100226GKWLSLLKHILKHAL-2/1112Not tested
371824176852YGRKKRRQRRRREADFFWSLCTADMSKilerFLIP26NA
37192387772I-C28H46N4O6, II-C27H44N4O6, III-C26H42N4O6Cepafungin complexNot AvailableNA
377322933412KKWβ2,2WKKc17IC50= 10±2 µMol/L
377422933412KW β2,2WKKc26IC50= 7.9±0.3 µMol/L
377522933412KK β2,2WKKc36IC50= 15±2 µMol/L
377622933412KW β2,2KKc45IC50= 12.6±0.6 µMol/L
377722933412KKW β2,2WKKc57IC50= 11±2 µMol/L
377822933412KW β2,2WKKc66IC50= 8±1 µMol/L
377922933412KK β2,2WKKc76IC50= 16±5 µMol/L
378022933412KW β2,2KKc85IC50= 20±2 µMol/L
378122933412KKWβ2,2WKKc17IC50= 22±5 µMol/L
378222933412KW β2,2WKKc26IC50= 1.71±0.6 µMol/L
378322933412KK β2,2WKKc36IC50= 92±2 µMol/L
378422933412KW β2,2KKc45IC50= 99±15 µMol/L
378522933412KKW β2,2WKKc57IC50= 23±3 µMol/L
378622933412KW β2,2WKKc66IC50= 26±2 µMol/L
378722933412KK β2,2WKKc76IC50= 157±30 µMol/L
378822933412KW β2,2KKc85IC50= 226±21 µMol/L
403012631273, 9266696GLFDVIKKVASVIGGLCitropin 1.116IC50= 5 M
403912631273, 9266696glfdvikkvasvigglCitropin 1.1D16IC50= 5 M
404812631273, 9266696GLFAVIKKVASVIGGL316IC50= 6 M
405712631273, 9266696GLFDVIKAVASVIGGL516IC50= 5 M
406612631273, 9266696GLFDVIKKVAAVIGGL716IC50= 5 M
407512631273, 9266696GLFDVIKKVASVIKGL1116IC50= 5 M
408412631273, 9266696GLFDVIKKVASVIKKL1316IC50= 5 M
409312631273, 9266696GLFDVIAKVASVIKKL1416IC50= 5 M
410212631273, 9266696GLFAVIKKVASVIKGL1516IC50= 5 M
411112631273, 9266696GLFAVIKKVASVIKKL1616IC50= 5 M
412012631273, 9266696GLFAVIKKVAAVIKKL1716IC50= 5 M
412912631273, 9266696GLFAVIKKVAAVIRRL1816IC50= 5 M
413812631273, 9266696GLFAVIKKVAKVIKKL1916IC50= 5 M
414712631273, 9266696GLFKVIKKVASVIGGL2216IC50= 5 M
415612631273, 9266696GLFKVIKKVAKVIKKL2316IC50= 5 M
416512631273, 9266696LGGIVSAVKKIVDFLGretro16IC50= 5 M
419915835725lwPsychrophilin D (1)Not AvailableID50=10.1 µg/ml
420815875779, 1429232Aoc-Hse-E-Dhb-Hyp-Hse-FLIILGLaxaphycin A12No inhibition at 4 µM
420915875779, 1429232Aoc-Hse-E-Dhb-Hyp-Hse-FLIILGLaxaphycin A12No inhibition at 4 µM
421015875779, 1429232Aoc-Hse-E-Dhb-Hyp-Hse-FLIILGLaxaphycin A12No inhibition at 4 µM
421115875779, 1429232A-Hleu-QN-MeIle-Hasn-TPLT-Ade-V-HleuLaxaphycin B1350% inhibition at 1 µM
421215875779, 1429232A-Hleu-QN-MeIle-Hasn-TPLT-Ade-V-HleuLaxaphycin B1344% inhibition at 1 µM
421315875779, 1429232A-Hleu-QN-MeIle-Hasn-TPLT-Ade-V-HleuLaxaphycin B1344% inhibition at 1 µM
421415875779, 1429232A-Hleu-QN-MeIle-Hasn-TPLT-Ade-V-HleuLaxaphycin B1344% inhibition at 1 µM
421515875779, 1429232A-Hleu-QN-MeIle-Hasn-TPLT-Ade-V-HleuLaxaphycin B1340% inhibition at 1 µM
421615875779, 1429232A-Hleu-QN-MeIle-Hasn-TPLT-Ade-V-HleuLaxaphycin B1340% inhibition at 1 µM
421715875779, 1429232A-Hleu-QN-MeIle-Hasn-TPLT-Ade-V-HleuLaxaphycin B1340% inhibition at 1 µM
446922076954IELLQARGGC-PemPeptide-110IC50 = 2.17 µM
447022076954IELLQARGGC-Pem-GGRRRRRRRRPeptide-210IC50 = 2.64 µM
447122076954RRRRRRRRGGC-PemPeptide-311IC50 = 6.24 µM
459221403917TRSSRAGLQFPVGRVHRLLRKBuforin 221IC50 =90-95 µg/ml
459321403917GLFDVIKKVASVIGGLCitropin 1.116IC50 =40 µg/ml
459421403917AKRHHGYKRKFHDemegen P-11312IC50 =85-90 µg/ml
459521403917ILRWPWWPWRRKOmiganan MBI-22612IC50 =80-85 µg/ml
459621403917GIGKFLKKAKKFGKAFVKILKKPexiganan MSI-7818IC50 =20-30 µg/ml
459721403917RGGRLCYCRRRFCVCVGRProtegrin 118IC50 =30-40 µg/ml
459821403917FLPLIGRVLSGILTemporin A13IC50 =80-90 µg/ml
461120802991CSSRTMHHCPeptide-209at 100 µM 90% viablity
46408445676VV-Nme-VPP-2-hydroxyisovaleryl-2-
oxo-4-methoxy-5-benzyl-3-pyrroline
Dolastatin 15Not AvailableIC50=.00013-.0013 nM
46418445676VV-Nme-VPP-2-hydroxyisovaleryl-2-
oxo-4-methoxy-5-benzyl-3-pyrroline
Dolastatin 15Not AvailableIC50=.00013-.0013 nM
46428445676VV-Nme-VPP-2-hydroxyisovaleryl-2-
oxo-4-methoxy-5-benzyl-3-pyrroline
Dolastatin 15Not AvailableIC50=.00013-.0013 nM
46438445676VV-Nme-VPP-2-hydroxyisovaleryl-2-
oxo-4-methoxy-5-benzyl-3-pyrroline
Dolastatin 15Not AvailableIC50=.00013-.0013 nM
464484456762-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-
[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-
(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-
1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-
dimethylbutanamide
Dolastatin 10Not AvailableIC50=.0013-.013 nM
464584456762-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-
[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-
(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-
1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-
dimethylbutanamide
Dolastatin 10Not AvailableIC50=.0013-.013 nM
464684456762-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-
[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-
(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-
1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-
dimethylbutanamide
Dolastatin 10Not AvailableIC50=.00013-.0013 nM
464784456762-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-
[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-
(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-
1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-
dimethylbutanamide
Dolastatin 10Not AvailableIC50=.0013-.013 nM
464823085771Not Available5a3IC50=10.6 µM
464923085771Not Available5b3IC50=7.1 µM
465023085771Not Available5c3IC50=4.1 µM
465123085771Not Available6a3IC50=14.4 µM
465223085771Not Available6b3IC50=11.0 µM
465323085771Not Available6c3IC50=4.3 µM
465423085771Not Available7a3IC50=>63 µM
465523085771Not Available7b3IC50=>78 µM
465623085771Not Available7c3IC50=79 µM
465723085771Not Available8a3IC50=136 µM
465823085771Not Available8b3IC50=>254 µM
465923085771Not Available8c3IC50=107 µM
466023085771Not Available9a3IC50=31 µM
466123085771Not Available9b3IC50=2.3 µM
466223085771Not Available9c3IC50=3.1 µM
466323085771Not Available10a3IC50=28 µM
466423085771Not Available10b3IC50=11.4 µM
466523085771Not Available10c3IC50=6.6 µM
466623085771Not Available11a3IC50=5.2 µM
466723085771Not Available11b3IC50=19 µM
466823085771Not Available11c3IC50=7.2 µM
466923085771Not Available12a3IC50=6.1 µM
467023085771Not Available12b3IC50=27 µM
467123085771Not Available12c3IC50=14 µM