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IDPMIDSEQUENCENAME LENGTHACTIVITY
1907NoneFALAFLAK-120B4LD50 =>1000 µg/ml
2059NoneFALAFLAK-120B4LD50 =>1000 µg/ml
2211NoneFALAFLAK-120B4LD50 =>1000 µg/ml
2363NoneFALAFLAK-120B4LD50 =>1000 µg/ml
2516NoneFALAFLAK-120B4LD50 =>1000 µg/ml
2659NoneFALAFLAK-120B4LD50 =>1000 µg/ml
2802NoneFALAFLAK-120B4LD50 = >1000 µg/ml
284515634655ERRPEGFR-related peptide430% Cell viability at 5 µg/ml
287223583573DEVDcaspase 3 inhibitor465% Cell viability at 20 µM
287323583573DEVDcaspase 3 inhibitor440% Cell viability at 30 µM
287423583573DEVDcaspase 3 inhibitor435 % Cell viability at 40 µM
318917787026(K-Aib-C(CH2CO-2'-Pac))2Dimer of peptide-paclitaxel conjugate3IC50 =1.31nM
319017787026(K-Aib-C(CH2CO-2'-Pac))3Dimer of peptide-paclitaxel conjugate3IC50 =2.85nM
319117787026(K-Aib-C(CH2CO-2'-Pac))4Dimer of peptide-paclitaxel conjugate3IC50 =0.62nM
319217787026(K-Aib-C(CH2CO-2'-Pac))3Trimer of peptide-paclitaxel conjugate3IC50 =1.70nM
319317787026(K-Aib-C(CH2CO-2'-Pac))3Trimer of peptide-paclitaxel conjugate3IC50 =3.88nM
319417787026(K-Aib-C(CH2CO-2'-Pac))3Trimer of peptide-paclitaxel conjugate3IC50 =3.00nM
319517787026(K-Aib-C(CH2CO-2'-Pac))4Tetramer of peptide-paclitaxel conjugate3IC50 =0.96nM
319617787026(K-Aib-C(CH2CO-2'-Pac))4Tetramer of peptide-paclitaxel conjugate3IC50 =1.30nM
319717787026(K-Aib-C(CH2CO-2'-Pac))4Tetramer of peptide-paclitaxel conjugate3IC50 =0.64nM
334223533710YPFPGβ-Casomorphins 5 f(60_64)4Inhibition at 9-11g/l
334522820149Structure GivenBAA-1Not AvailableIC50 = 8.1 µg/ml
334622820149Structure GivenBAA-2Not AvailableIC50 = 3.8 µg/ml
334711943716Not AvailableHα-Defensin HNPs-1Not AvailableInhibition at 12.5 µg/ml
334811943716Not AvailableHα-Defensin HNPs-2Not AvailableInhibition at 12.5 µg/ml
334911943716Not AvailableHα-Defensin HNPs-3Not AvailableInhibition at 12.5 µg/ml
37192387772I-C28H46N4O6, II-C27H44N4O6, III-C26H42N4O6Cepafungin complexNot AvailableNA
384716722632YA*8214.2% inhibition at 10-6
384816722632YA*8219.7% inhibition at 10-5
384916722632YA*8224.9% inhibition at 10-4
385016722632YA*8230.4% inhibition at 10-3
385116722632YA*8210% inhibition at 10-5
385216722632YA*828.2% inhibition at 10-4
385316722632YA*8236.1% inhibition at 10-3
385416722632YA*826.5% inhibition at 10-6
385516722632YA*8214% inhibition at 10-5
385616722632YA*827.5% inhibition at 10-4
385716722632YA*8214% inhibition at 10-3
385816722632YA*829.8% inhibition at 10-6
385916722632YA*821.6% inhibition at 10-5
386016722632YA*825.4% inhibition at 10-4
386116722632YA*8226.5% inhibition at 10-3
386216722632YA*8212.9% inhibition at 10-6
386316722632YA*8216.5% inhibition at 10-5
386416722632YA*8228.1% inhibition at 10-4
386516722632YA*8258.2% inhibition at 10-3
386616722632YA*823.5% inhibition at 10-6
386716722632YA*8222.7% inhibition at 10-5
386816722632YA*8218.9% inhibition at 10-4
386916722632YA*8226.4% inhibition at 10-3
387016722632YA*822.4% inhibition at 10-5
387116722632YA*827.5% inhibition at 10-4
387216722632YSA*936.2% inhibition at 10-6
387316722632YSA*936.4% inhibition at 10-5
387416722632YSA*938.2% inhibition at 10-4
387516722632YSA*9321.2% inhibition at 10-3
387616722632YSA*937.5% inhibition at 10-6
387716722632YSA*936.1% inhibition at 10-5
387816722632YSA*933.1% inhibition at 10-4
387916722632YSA*9314.8% inhibition at 10-3
388016722632YSA*933.9% inhibition at 10-5
388116722632YSA*937.3% inhibition at 10-3
388216722632YSA*934.9% inhibition at 10-6
388316722632YSA*938.9% inhibition at 10-5
388416722632YSA*933.4% inhibition at 10-4
388516722632YSA*9320.8% inhibition at 10-3
388616722632YSA*9310.5% inhibition at 10-6
388716722632YSA*9321.9% inhibition at 10-5
388816722632YSA*9311.8% inhibition at 10-4
388916722632YSA*9317.9% inhibition at 10-3
389016722632YSA*933.7% inhibition at 10-6
389116722632YSA*9316.5% inhibition at 10-5
389216722632YSA*938.4% inhibition at 10-4
389316722632YSA*9314.5% inhibition at 10-3
389416722632YSA*931.1% inhibition at 10-5
389516722632YSA*931.2% inhibition at 10-4
389616722632YSA*9317.8% inhibition at 10-3
389716722632YSA*1038.5% inhibition at 10-6
389816722632YSA*1034.9% inhibition at 10-5
389916722632YSA*1031.9% inhibition at 10-4
390016722632YSA*10316.2% inhibition at 10-3
390116722632YSA*1037.2% inhibition at 10-6
390216722632YSA*10317.1% inhibition at 10-5
390316722632YSA*10311.0% inhibition at 10-4
390416722632YSA*10320.5% inhibition at 10-3
390516722632YSA*1033.0% inhibition at 10-6
390616722632YSA*1034.7% inhibition at 10-5
390716722632YSA*1032.7% inhibition at 10-4
390816722632YSA*1037.3% inhibition at 10-3
390916722632YSA*1030.7% inhibition at 10-6
391016722632YSA*1038.3% inhibition at 10-5
391116722632YSA*10310.5% inhibition at 10-4
391216722632YSA*10321.8% inhibition at 10-3
391316722632YSA*10310.7% inhibition at 10-6
391416722632YSA*10310.0% inhibition at 10-5
391516722632YSA*1037.7% inhibition at 10-4M
391616722632YSA*10318.7% inhibition at 10-3M
391716722632YSA*G1542.7% inhibition at 10-6M
391816722632YSA*G1542.0% inhibition at 10-5M
391916722632YSA*G15418.8% inhibition at 10-4M
392016722632YSA*G15426.7% inhibition at 10-3M
392116722632YSA*G1549.8% inhibition at 10-6M
392216722632YSA*G1547.3% inhibition at 10-5M
392316722632YSA*G1549.9% inhibition at 10-4M
392416722632YSA*G15428.2% inhibition at 10-3M
392516722632YSA*G1541.6% inhibition at 10-6M
392616722632YSA*G1542.9% inhibition at 10-5M
392716722632YSA*G1545.9% inhibition at 10-4M
392816722632YSA*G15417.9% inhibition at 10-3M
392916722632YSA*G1545.4% inhibition at 10-6M
393016722632YSA*G1547.4% inhibition at 10-5M
393116722632YSA*G1549.5% inhibition at 10-4M
393216722632YSA*G15415.7% inhibition at 10-3M
393316722632YSA*G15413.6% inhibition at 10-6M
393416722632YSA*G15420.4% inhibition at 10-5M
393516722632YSA*G15414.4% inhibition at 10-4M
393616722632YSA*G15423.4% inhibition at 10-3M
393716722632YSA*G1542.2% inhibition at 10-6M
393816722632YSA*G1544.2% inhibition at 10-5M
393916722632YSA*G1546.4% inhibition at 10-4M
394016722632YSA*G1546.2% inhibition at 10-3M
394116722632YSA*G15421.2% inhibition at 10-3M
394216722632YRA*G1644.6% inhibition at 10-6M
394316722632YRA*G1644.9% inhibition at 10-5M
394416722632YRA*G16412.6% inhibition at 10-4M
394516722632YRA*G16426.4% inhibition at 10-3M
394616722632YRA*G16411.0% inhibition at 10-6M
394716722632YRA*G16411.7% inhibition at 10-5M
394816722632YRA*G16411.6% inhibition at 10-4M
394916722632YRA*G16428.2% inhibition at 10-3M
395016722632YRA*G1641.2% inhibition at 10-5M
395116722632YRA*G1643.3% inhibition at 10-4M
395216722632YRA*G16419.4% inhibition at 10-3M
395316722632YRA*G1647.6% inhibition at 10-6M
395416722632YRA*G1643.8% inhibition at 10-5M
395516722632YRA*G16412.4% inhibition at 10-4M
395616722632YRA*G16422.4% inhibition at 10-3M
395716722632YRA*G16417.0% inhibition at 10-6M
395816722632YRA*G16413.5% inhibition at 10-5M
395916722632YRA*G16413.5% inhibition at 10-4M
396016722632YRA*G16425.3% inhibition at 10-3M
396116722632YRA*G1648.1% inhibition at 10-6M
396216722632YRA*G1646.9% inhibition at 10-5M
396316722632YRA*G1648.1% inhibition at 10-4M
396416722632YRA*G1648.6% inhibition at 10-3M
396516722632YRA*G16415.6% inhibition at 10-3M
419915835725lwPsychrophilin D (1)Not AvailableID50=10.1 µg/ml
421815887970Not AvailableSansalv amide ANot AvailableEC50=7.5 µM
421916091933YSLTyroserleutide349.4% cytotoxic at 0.1 µg/ml
422016091933YSLTyroserleutide351.2% cytotoxic at 1 µg/ml
422116091933YSLTyroserleutide353.0% cytotoxic at 10 µg/ml
422216091933YSLTyroserleutide361.2% cytotoxic at 100 µg/ml
422316091933YSLTyroserleutide339.0% cytotoxic at 0.1 µg/ml
422416091933YSLTyroserleutide320.8% cytotoxic at 1 µg/ml
422516091933YSLTyroserleutide333.8% cytotoxic at 10 µg/ml
422616091933YSLTyroserleutide335.6% cytotoxic at 100 µg/ml
46408445676VV-Nme-VPP-2-hydroxyisovaleryl-2-
oxo-4-methoxy-5-benzyl-3-pyrroline
Dolastatin 15Not AvailableIC50=.00013-.0013 nM
46418445676VV-Nme-VPP-2-hydroxyisovaleryl-2-
oxo-4-methoxy-5-benzyl-3-pyrroline
Dolastatin 15Not AvailableIC50=.00013-.0013 nM
46428445676VV-Nme-VPP-2-hydroxyisovaleryl-2-
oxo-4-methoxy-5-benzyl-3-pyrroline
Dolastatin 15Not AvailableIC50=.00013-.0013 nM
46438445676VV-Nme-VPP-2-hydroxyisovaleryl-2-
oxo-4-methoxy-5-benzyl-3-pyrroline
Dolastatin 15Not AvailableIC50=.00013-.0013 nM
464484456762-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-
[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-
(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-
1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-
dimethylbutanamide
Dolastatin 10Not AvailableIC50=.0013-.013 nM
464584456762-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-
[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-
(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-
1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-
dimethylbutanamide
Dolastatin 10Not AvailableIC50=.0013-.013 nM
464684456762-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-
[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-
(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-
1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-
dimethylbutanamide
Dolastatin 10Not AvailableIC50=.00013-.0013 nM
464784456762-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-
[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-
(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-
1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-
dimethylbutanamide
Dolastatin 10Not AvailableIC50=.0013-.013 nM
464823085771Not Available5a3IC50=10.6 µM
464923085771Not Available5b3IC50=7.1 µM
465023085771Not Available5c3IC50=4.1 µM
465123085771Not Available6a3IC50=14.4 µM
465223085771Not Available6b3IC50=11.0 µM
465323085771Not Available6c3IC50=4.3 µM
465423085771Not Available7a3IC50=>63 µM
465523085771Not Available7b3IC50=>78 µM
465623085771Not Available7c3IC50=79 µM
465723085771Not Available8a3IC50=136 µM
465823085771Not Available8b3IC50=>254 µM
465923085771Not Available8c3IC50=107 µM
466023085771Not Available9a3IC50=31 µM
466123085771Not Available9b3IC50=2.3 µM
466223085771Not Available9c3IC50=3.1 µM
466323085771Not Available10a3IC50=28 µM
466423085771Not Available10b3IC50=11.4 µM
466523085771Not Available10c3IC50=6.6 µM
466623085771Not Available11a3IC50=5.2 µM
466723085771Not Available11b3IC50=19 µM
466823085771Not Available11c3IC50=7.2 µM
466923085771Not Available12a3IC50=6.1 µM
467023085771Not Available12b3IC50=27 µM
467123085771Not Available12c3IC50=14 µM
467594928452-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-
[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-
1-(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-1-
yl]-5-methyl-1-oxoheptan-4-yl]-N,3-dimethylbutanamide
Dolastatin 10Not AvailableIC50=0.5 nM