Detail description

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3823 details
Primary information
CancerPPD ID3823
PMID22963485
YEAR2012
SEQUENCEMNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANNF
VLIVSQLQPSQENEMFSIRGDSAHRRFLLFRRAFK
QLDVEAALTKALGEVDILLTWMQKFYKL
LENGTH207
NAMERGD-mda-7
C-ter ModificationFree
N-ter ModificationFree
Linear/CyclicLinear
L/D/MixL
Non-NaturalNone
NATUREAnticancer
ACTIVITYApoptotic rate(%)= >70% at concentration of 8 µg/ml
SOURCEDerived from wtmda-7/IL-24 by insertion og a glycine residue between Arg(164) and Asp(165).
ASSAYMTT assay
CELL LINEMCF-7
TEST TIME72-h
Secondary information
STRUCTURE
Predicted Structure
DSSP statesCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCSCCEEETTEEECCCCHHHHHHHHHHHHHHHHHHCCCTTCCSSCCCCSSCSSHHHHHHHHHHHHHHHHHTHHHHSCCSSSCHHHHHHHHHHHHHHHHHHHHHTTTTTTSSCCCCTTHHHHHHHHHHHHHHHSCHHHHHHHHHHTHHHHHHSSSSSCCC
SMILES
External Links
PDB exactPDB partialSP exactSP partialTrEMBL exactTrEMBL partialIEDB exactIEDB partial
NANANANANANANANA