Epidermal Growth Factor Receptor Inhibitor Database
Activity against kinases
Molecule Id: EGIN0000003
S.No.
Kinase
Mutant
IC
50
K
i
K
d
Enz. inhib. (%)
Inhib. Conc.
Cellular IC
50
Cell line
Growth Factor
1
BT474
-
80 nM
-
-
-
-
-
-
-
2
BT474
-
100 nM
-
-
-
-
-
-
-
3
BT474
-
100 nM
-
-
-
-
-
-
-