Epidermal Growth Factor Receptor Inhibitor Database
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| Activity against kinases | ||||||||||||||
| Molecule Id: EGIN0000232 | ||||||||||||||
| S.No. | Kinase | Mutant | IC50 | Ki | Kd | Enz. inhib. (%) | Inhib. Conc. | Cellular IC50 | Cell line | Growth Factor | ||||
| 1 | Insulin receptor | Purified protein kinase | >50000 nM | - | - | - | - | - | - | - | ||||
| 2 | PDGFr | Purified protein kinase | >50000 nM | - | - | - | - | - | - | - | ||||
| 3 | PKC | Purified protein kinase | >50000 nM | - | - | - | - | - | - | - | ||||
| 4 | Insulin receptor | Receptor phosphorylation in fibroblasts | >50000 nM | - | - | - | - | - | - | - | ||||
| 5 | PDGFr | Receptor phosphorylation in fibroblasts | >50000 nM | - | - | - | - | - | - | - | ||||