Epidermal Growth Factor Receptor Inhibitor Database


Activity against kinases
Molecule Id: EGIN0000232
S.No. Kinase Mutant IC50 Ki Kd Enz. inhib. (%) Inhib. Conc. Cellular IC50 Cell line Growth Factor
1PDGFrPurified protein kinase>50000 nM-------
2PDGFrReceptor phosphorylation in fibroblasts>50000 nM-------