Epidermal Growth Factor Receptor Inhibitor Database
Activity against kinases
Molecule Id: EGIN0001486
S.No.
Kinase
Mutant
IC
50
K
i
K
d
Enz. inhib. (%)
Inhib. Conc.
Cellular IC
50
Cell line
Growth Factor
1
VEGFR2
-
30000nM
-
-
-
-
-
-
-
2
SRC
-
82000nM
-
-
-
-
-
-
-
3
TIE2
-
95000nM
-
-
-
-
-
-
-