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| Activity against kinases | ||||||||||||||
| Molecule Id: EGIN0002336 | ||||||||||||||
| S.No. | Kinase | Mutant | IC50 | Ki | Kd | Enz. inhib. (%) | Inhib. Conc. | Cellular IC50 | Cell line | Growth Factor | ||||
| 1 | VEGFR2 | - | >200000nM | - | - | - | - | - | - | - | ||||
| 2 | PDGFR beta | - | >500000nM | - | - | - | - | - | - | - | ||||
| 3 | DHFR human | - | 86500nM | - | - | - | - | - | - | - | ||||