Epidermal Growth Factor Receptor Inhibitor Database
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| Activity against kinases | ||||||||||||||
| Molecule Id: EGIN0002635 | ||||||||||||||
| S.No. | Kinase | Mutant | IC50 | Ki | Kd | Enz. inhib. (%) | Inhib. Conc. | Cellular IC50 | Cell line | Growth Factor | ||||
| 1 | CDK4/Cyc | - | 1000000nM | - | - | - | - | - | - | - | ||||
| 2 | CDK2/CycE | - | 1500nM | - | - | - | - | - | - | - | ||||
| 3 | PKC | - | 160000nM | - | - | - | - | - | - | - | ||||
| 4 | PKA | - | 260000nM | - | - | - | - | - | - | - | ||||
| 5 | CDK1/CycB1 | - | 600nM | - | - | - | - | - | - | - | ||||
| 6 | MAP | - | 94000nM | - | - | - | - | - | - | - | ||||