Epidermal Growth Factor Receptor Inhibitor Database


Activity against kinases
Molecule Id: EGIN0004339
S.No. Kinase Mutant IC50 Ki Kd Enz. inhib. (%) Inhib. Conc. Cellular IC50 Cell line Growth Factor
1Lck%ACTIVITY RELATIVE TO 100%DMSO---110 然---
2YES1%ACTIVITY RELATIVE TO 100%DMSO---410 然---
3EPH-B3%ACTIVITY RELATIVE TO 100%DMSO---510 然---
4RIPK2%ACTIVITY RELATIVE TO 100%DMSO---1010 然---
5MINK1%ACTIVITY RELATIVE TO 100%DMSO---1210 然---
6Src%ACTIVITY RELATIVE TO 100%DMSO---1310 然---
7PKD1%ACTIVITY RELATIVE TO 100%DMSO---1410 然---
8MNK2%ACTIVITY RELATIVE TO 100%DMSO---2110 然---
9MELK%ACTIVITY RELATIVE TO 100%DMSO---2510 然---
10EPH-A2%ACTIVITY RELATIVE TO 100%DMSO---2610 然---
11PHK%ACTIVITY RELATIVE TO 100%DMSO---2610 然---
12CHK2%ACTIVITY RELATIVE TO 100%DMSO---2710 然---
13CAMK1%ACTIVITY RELATIVE TO 100%DMSO---3010 然---
14GCK%ACTIVITY RELATIVE TO 100%DMSO---3010 然---
15p38a%ACTIVITY RELATIVE TO 100%DMSO---3010 然---
16FGF-R1%ACTIVITY RELATIVE TO 100%DMSO---3110 然---
17DYRK3%ACTIVITY RELATIVE TO 100%DMSO---3210 然---
18AuroraB%ACTIVITY RELATIVE TO 100%DMSO---3310 然---
19BRSK2%ACTIVITY RELATIVE TO 100%DMSO---3610 然---
20BTK%ACTIVITY RELATIVE TO 100%DMSO---3610 然---
21PRK2%ACTIVITY RELATIVE TO 100%DMSO---3610 然---
22VEGFR%ACTIVITY RELATIVE TO 100%DMSO---3610 然---
23NUAK1%ACTIVITY RELATIVE TO 100%DMSO---3710 然---
24CK1%ACTIVITY RELATIVE TO 100%DMSO---4410 然---
25MKK1%ACTIVITY RELATIVE TO 100%DMSO---4510 然---
26BRSK1%ACTIVITY RELATIVE TO 100%DMSO---4610 然---
27PIM1%ACTIVITY RELATIVE TO 100%DMSO---4610 然---
28SmMLCK%ACTIVITY RELATIVE TO 100%DMSO---4810 然---
29JNK1%ACTIVITY RELATIVE TO 100%DMSO---4910 然---
30JNK2%ACTIVITY RELATIVE TO 100%DMSO---5010 然---
31DYRK2%ACTIVITY RELATIVE TO 100%DMSO---5210 然---
32SYK%ACTIVITY RELATIVE TO 100%DMSO---5710 然---
33PKBb%ACTIVITY RELATIVE TO 100%DMSO---6110 然---
34IKKB%ACTIVITY RELATIVE TO 100%DMSO---6210 然---
35JNK3%ACTIVITY RELATIVE TO 100%DMSO---6210 然---
36p38b%ACTIVITY RELATIVE TO 100%DMSO---6310 然---
37MetNK1%ACTIVITY RELATIVE TO 100%DMSO---6410 然---
38PIM3%ACTIVITY RELATIVE TO 100%DMSO---6610 然---
39PAK5%ACTIVITY RELATIVE TO 100%DMSO---6810 然---
40IRAK4%ACTIVITY RELATIVE TO 100%DMSO---7010 然---
41IGF-1R%ACTIVITY RELATIVE TO 100%DMSO---7110 然---
42MAPKAP-K3%ACTIVITY RELATIVE TO 100%DMSO---7210 然---
43CSK%ACTIVITY RELATIVE TO 100%DMSO---7310 然---
44CAMKKb%ACTIVITY RELATIVE TO 100%DMSO---7410 然---
45RSK2%ACTIVITY RELATIVE TO 100%DMSO---7410 然---
46MARK4%ACTIVITY RELATIVE TO 100%DMSO---7510 然---
47PIM2%ACTIVITY RELATIVE TO 100%DMSO---7510 然---
48SRPK1%ACTIVITY RELATIVE TO 100%DMSO---7510 然---
49p38d%ACTIVITY RELATIVE TO 100%DMSO---7610 然---
50MARK2%ACTIVITY RELATIVE TO 100%DMSO---7710 然---
51PDK1%ACTIVITY RELATIVE TO 100%DMSO---7810 然---
52IRR%ACTIVITY RELATIVE TO 100%DMSO---7910 然---
53MLK1%ACTIVITY RELATIVE TO 100%DMSO---7910 然---
54PAK2%ACTIVITY RELATIVE TO 100%DMSO---7910 然---
55PAK4%ACTIVITY RELATIVE TO 100%DMSO---7910 然---
56MST4%ACTIVITY RELATIVE TO 100%DMSO---8010 然---
57MST2%ACTIVITY RELATIVE TO 100%DMSO---8110 然---
58PKCa%ACTIVITY RELATIVE TO 100%DMSO---8210 然---
59SGK1%ACTIVITY RELATIVE TO 100%DMSO---8210 然---
60CHK1%ACTIVITY RELATIVE TO 100%DMSO---8310 然---
61ERK1%ACTIVITY RELATIVE TO 100%DMSO---8310 然---
62PAK6%ACTIVITY RELATIVE TO 100%DMSO---8310 然---
63AMPK%ACTIVITY RELATIVE TO 100%DMSO---8410 然---
64MLK3%ACTIVITY RELATIVE TO 100%DMSO---8410 然---
65PRAK%ACTIVITY RELATIVE TO 100%DMSO---8410 然---
66TBK1%ACTIVITY RELATIVE TO 100%DMSO---8410 然---
67DYRK1A%ACTIVITY RELATIVE TO 100%DMSO---8510 然---
68ERK8%ACTIVITY RELATIVE TO 100%DMSO---8510 然---
69IR-HIS%ACTIVITY RELATIVE TO 100%DMSO---8510 然---
70NEK6%ACTIVITY RELATIVE TO 100%DMSO---8510 然---
71TTK%ACTIVITY RELATIVE TO 100%DMSO---8510 然---
72MAPKAP-K2%ACTIVITY RELATIVE TO 100%DMSO---8610 然---
73PKA%ACTIVITY RELATIVE TO 100%DMSO---8610 然---
74PKCz%ACTIVITY RELATIVE TO 100%DMSO---8610 然---
75S6K1%ACTIVITY RELATIVE TO 100%DMSO---8710 然---
76AuroraA%ACTIVITY RELATIVE TO 100%DMSO---8810 然---
77CDK2-CycA%ACTIVITY RELATIVE TO 100%DMSO---8810 然---
78ERK2%ACTIVITY RELATIVE TO 100%DMSO---8810 然---
79ROCK2%ACTIVITY RELATIVE TO 100%DMSO---8810 然---
80GSK3b%ACTIVITY RELATIVE TO 100%DMSO---8910 然---
81RSK1%ACTIVITY RELATIVE TO 100%DMSO---8910 然---
82CK2%ACTIVITY RELATIVE TO 100%DMSO---9010 然---
83IKKe%ACTIVITY RELATIVE TO 100%DMSO---9210 然---
84LKB1%ACTIVITY RELATIVE TO 100%DMSO---9410 然---
85MARK3%ACTIVITY RELATIVE TO 100%DMSO---9410 然---
86p38g%ACTIVITY RELATIVE TO 100%DMSO---9410 然---
87NEK2a%ACTIVITY RELATIVE TO 100%DMSO---9510 然---
88HIPK3%ACTIVITY RELATIVE TO 100%DMSO---9610 然---
89MSK1%ACTIVITY RELATIVE TO 100%DMSO---9610 然---
90EF2K%ACTIVITY RELATIVE TO 100%DMSO---9910 然---
91PKBa%ACTIVITY RELATIVE TO 100%DMSO---10010 然---
92HIPK1%ACTIVITY RELATIVE TO 100%DMSO---10310 然---
93HIPK2%ACTIVITY RELATIVE TO 100%DMSO---10410 然---
94PLK1%ACTIVITY RELATIVE TO 100%DMSO---10910 然---