Epidermal Growth Factor Receptor Inhibitor Database


Activity against kinases
Molecule Id: EGIN0004340
S.No. Kinase Mutant IC50 Ki Kd Enz. inhib. (%) Inhib. Conc. Cellular IC50 Cell line Growth Factor
1Lck%ACTIVITY RELATIVE TO 100%DMSO---310 然---
2YES1%ACTIVITY RELATIVE TO 100%DMSO---710 然---
3PHK%ACTIVITY RELATIVE TO 100%DMSO---1010 然---
4RIPK2%ACTIVITY RELATIVE TO 100%DMSO---1010 然---
5PIM1%ACTIVITY RELATIVE TO 100%DMSO---1210 然---
6MNK2%ACTIVITY RELATIVE TO 100%DMSO---1410 然---
7EPH-B3%ACTIVITY RELATIVE TO 100%DMSO---1710 然---
8PKD1%ACTIVITY RELATIVE TO 100%DMSO---1810 然---
9SmMLCK%ACTIVITY RELATIVE TO 100%DMSO---1810 然---
10AuroraB%ACTIVITY RELATIVE TO 100%DMSO---2110 然---
11DYRK3%ACTIVITY RELATIVE TO 100%DMSO---2710 然---
12BRSK2%ACTIVITY RELATIVE TO 100%DMSO---2910 然---
13MKK1%ACTIVITY RELATIVE TO 100%DMSO---2910 然---
14PIM3%ACTIVITY RELATIVE TO 100%DMSO---3210 然---
15MINK1%ACTIVITY RELATIVE TO 100%DMSO---3510 然---
16FGF-R1%ACTIVITY RELATIVE TO 100%DMSO---3710 然---
17PRK2%ACTIVITY RELATIVE TO 100%DMSO---3710 然---
18CHK2%ACTIVITY RELATIVE TO 100%DMSO---3810 然---
19NUAK1%ACTIVITY RELATIVE TO 100%DMSO---3910 然---
20Src%ACTIVITY RELATIVE TO 100%DMSO---4410 然---
21GCK%ACTIVITY RELATIVE TO 100%DMSO---4810 然---
22MELK%ACTIVITY RELATIVE TO 100%DMSO---4910 然---
23MetNK1%ACTIVITY RELATIVE TO 100%DMSO---4910 然---
24VEGFR%ACTIVITY RELATIVE TO 100%DMSO---5010 然---
25DYRK2%ACTIVITY RELATIVE TO 100%DMSO---5110 然---
26BRSK1%ACTIVITY RELATIVE TO 100%DMSO---5210 然---
27EPH-A2%ACTIVITY RELATIVE TO 100%DMSO---5310 然---
28CAMK1%ACTIVITY RELATIVE TO 100%DMSO---5710 然---
29PIM2%ACTIVITY RELATIVE TO 100%DMSO---6210 然---
30CSK%ACTIVITY RELATIVE TO 100%DMSO---6310 然---
31p38a%ACTIVITY RELATIVE TO 100%DMSO---6310 然---
32AMPK%ACTIVITY RELATIVE TO 100%DMSO---6510 然---
33DYRK1A%ACTIVITY RELATIVE TO 100%DMSO---6510 然---
34MLK3%ACTIVITY RELATIVE TO 100%DMSO---6510 然---
35AuroraA%ACTIVITY RELATIVE TO 100%DMSO---6610 然---
36CAMKKb%ACTIVITY RELATIVE TO 100%DMSO---6610 然---
37CK1%ACTIVITY RELATIVE TO 100%DMSO---6610 然---
38SYK%ACTIVITY RELATIVE TO 100%DMSO---6710 然---
39ERK1%ACTIVITY RELATIVE TO 100%DMSO---7010 然---
40IRR%ACTIVITY RELATIVE TO 100%DMSO---7010 然---
41PKCa%ACTIVITY RELATIVE TO 100%DMSO---7210 然---
42RSK1%ACTIVITY RELATIVE TO 100%DMSO---7210 然---
43MARK4%ACTIVITY RELATIVE TO 100%DMSO---7410 然---
44PAK2%ACTIVITY RELATIVE TO 100%DMSO---7510 然---
45S6K1%ACTIVITY RELATIVE TO 100%DMSO---7510 然---
46TBK1%ACTIVITY RELATIVE TO 100%DMSO---7510 然---
47JNK1%ACTIVITY RELATIVE TO 100%DMSO---7610 然---
48JNK2%ACTIVITY RELATIVE TO 100%DMSO---7710 然---
49NEK6%ACTIVITY RELATIVE TO 100%DMSO---7710 然---
50ERK8%ACTIVITY RELATIVE TO 100%DMSO---7810 然---
51MST2%ACTIVITY RELATIVE TO 100%DMSO---7810 然---
52RSK2%ACTIVITY RELATIVE TO 100%DMSO---7810 然---
53BTK%ACTIVITY RELATIVE TO 100%DMSO---7910 然---
54CHK1%ACTIVITY RELATIVE TO 100%DMSO---7910 然---
55IR-HIS%ACTIVITY RELATIVE TO 100%DMSO---7910 然---
56p38d%ACTIVITY RELATIVE TO 100%DMSO---7910 然---
57PAK6%ACTIVITY RELATIVE TO 100%DMSO---7910 然---
58JNK3%ACTIVITY RELATIVE TO 100%DMSO---8010 然---
59PKBb%ACTIVITY RELATIVE TO 100%DMSO---8010 然---
60IRAK4%ACTIVITY RELATIVE TO 100%DMSO---8110 然---
61MAPKAP-K3%ACTIVITY RELATIVE TO 100%DMSO---8110 然---
62p38b%ACTIVITY RELATIVE TO 100%DMSO---8110 然---
63MARK2%ACTIVITY RELATIVE TO 100%DMSO---8210 然---
64PAK4%ACTIVITY RELATIVE TO 100%DMSO---8310 然---
65PAK5%ACTIVITY RELATIVE TO 100%DMSO---8410 然---
66p38g%ACTIVITY RELATIVE TO 100%DMSO---8510 然---
67MARK3%ACTIVITY RELATIVE TO 100%DMSO---8610 然---
68PKCz%ACTIVITY RELATIVE TO 100%DMSO---8610 然---
69TTK%ACTIVITY RELATIVE TO 100%DMSO---8610 然---
70MLK1%ACTIVITY RELATIVE TO 100%DMSO---8710 然---
71SRPK1%ACTIVITY RELATIVE TO 100%DMSO---8710 然---
72ERK2%ACTIVITY RELATIVE TO 100%DMSO---8810 然---
73MST4%ACTIVITY RELATIVE TO 100%DMSO---8810 然---
74PDK1%ACTIVITY RELATIVE TO 100%DMSO---8810 然---
75IKKe%ACTIVITY RELATIVE TO 100%DMSO---8910 然---
76PRAK%ACTIVITY RELATIVE TO 100%DMSO---8910 然---
77IKKB%ACTIVITY RELATIVE TO 100%DMSO---9010 然---
78MAPKAP-K2%ACTIVITY RELATIVE TO 100%DMSO---9010 然---
79EF2K%ACTIVITY RELATIVE TO 100%DMSO---9110 然---
80PKA%ACTIVITY RELATIVE TO 100%DMSO---9110 然---
81CDK2-CycA%ACTIVITY RELATIVE TO 100%DMSO---9310 然---
82MSK1%ACTIVITY RELATIVE TO 100%DMSO---9310 然---
83SGK1%ACTIVITY RELATIVE TO 100%DMSO---9310 然---
84PLK1%ACTIVITY RELATIVE TO 100%DMSO---9510 然---
85ROCK2%ACTIVITY RELATIVE TO 100%DMSO---9510 然---
86CK2%ACTIVITY RELATIVE TO 100%DMSO---9610 然---
87GSK3b%ACTIVITY RELATIVE TO 100%DMSO---9610 然---
88HIPK2%ACTIVITY RELATIVE TO 100%DMSO---9710 然---
89NEK2a%ACTIVITY RELATIVE TO 100%DMSO---9710 然---
90LKB1%ACTIVITY RELATIVE TO 100%DMSO---10310 然---
91PKBa%ACTIVITY RELATIVE TO 100%DMSO---10310 然---
92IGF-1R%ACTIVITY RELATIVE TO 100%DMSO---10510 然---
93HIPK3%ACTIVITY RELATIVE TO 100%DMSO---10610 然---
94HIPK1%ACTIVITY RELATIVE TO 100%DMSO---12610 然---