Epidermal Growth Factor Receptor Inhibitor Database
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| Activity against kinases | ||||||||||||||
| Molecule Id: EGIN0004465 | ||||||||||||||
| S.No. | Kinase | Mutant | IC50 | Ki | Kd | Enz. inhib. (%) | Inhib. Conc. | Cellular IC50 | Cell line | Growth Factor | ||||
| 1 | PDGFR-alpha | - | - | - | - | 18.70% | 50 µM | - | - | - | ||||
| 2 | PDGFR-beta | - | - | - | - | 17.80% | 50 µM | - | - | - | ||||
| 3 | VEGFR-2(KDR) | - | - | - | - | 16.50% | 50 µM | - | - | - | ||||
| 4 | PI3K-a | - | - | - | - | 3.70% | 50 µM | - | - | - | ||||