ID SEQ Non-natural-modification 1020 GW*LR**K**AAK**SVGK**FY*Y*K**HK*Y*Y*IK*AAWQIGKHAL W*=6-bromotryptophan,R**=dihydroxyarginine, Y* = 3,4-dihydroxyphenylalanine,K* = 5-hydroxylysine, K**= dihydroxylysine 1021 GW*LR**K**AAK**SVGK**FY*Y*K**HK*Y*Y*IK*AAWQIGKHAL W*=6-bromotryptophan,R**=dihydroxyarginine, Y* = 3,4-dihydroxyphenylalanine,K* = 5-hydroxylysine, K**= dihydroxylysine 1091 APC-L-ACPC-K-ACPC-L-APC-L-ACPC-K-ACPC-L-APC-L-ACPC APC and ACPC 1092 APC-L-ACPC-L-APC-L-ACPC-K-ACPC-L-ACPC-K-ACPC-L-APC APC and ACPC 1093 ACPC-L-APC-K-APC-L-ACPC-K-APC-L-ACPC-L-ACPC-L-ACPC APC and ACPC 1094 APC-L-APC-L-ACPC-K-ACPC-L-ACPC-L-APC-L-ACPC-K-ACPC APC and ACPC 1095 APC-L-ACPC-L-APC-L-ACPC-L-APC-L-ACPC-K-ACPC-L-APC APC and ACPC 1096 APC-F-ACPC-L-APC-L-ACPC-F-APC-F-ACPC-K-ACPC-L-APC APC and ACPC 1097 APC-L-ACPC-K-ACPC-A-APC-A-ACPC-K-ACPC-A-APC-L-ACPC APC and ACPC 1098 APC-L-ACPC-A-APC-A-ACPC-K-ACPC-L-ACPC-K-ACPC-A-APC APC and ACPC 1099 ACPC-A-APC-K-APC-L-ACPC-K-APC-A-ACPC-A-ACPC-L-ACPC APC and ACPC 1125 KWKLFKK-ΔF-GAVLKVL ΔF = α, β-dehydrophenylalanine (ΔPhe) 1126 KWKL-ΔF-KKIGAV-ΔF-KVL ΔF = α, β-dehydrophenylalanine (ΔPhe) 1127 KWKL-ΔF-KK-ΔF-GAV-ΔF-KVL ΔF = α, β-dehydrophenylalanine (ΔPhe) 1157 GIINTLQKYYCRVRGGRCAVLSCLPKEEQIGKCSTRGRKCCRRKK Cystein is protected by Acm 1292 Aib-GL-Aib-GGL-Aib-GI Aib (α-aminoisobutyric acid) 1293 Aib-GL-Aib-GGL-Aib-GIL Aib (α-aminoisobutyric acid) 1294 Aib-GGL-Aib-GIL Aib (α-aminoisobutyric acid) 1295 Aib-GIL Aib (α-aminoisobutyric acid) 1464 G-ΔF-RK-ΔF-HK-ΔF-WA ΔF=α,β-didehydrophenylalanine 1465 G-ΔF-RK-ΔF-KA-ΔF-WH ΔF=α,β-didehydrophenylalanine 1508 GFLSILKKVLPKV-Met(O)-AH-Met(O)-K Met (O)= methionine sulfoxide 1509 GFLSILKKVLPKV-Met(O2)-AH-Met(O2)-K Met (O2)=methionine sulfone 1510 GFLSILKKVLPKV-Nle-AH-Nle-K Nle= norleucine 1511 GFLSILKKVLPKV-Met-AH-Nle-K Nle= norleucine 1512 GFLSILKKVLPKV-Nle-AH-Met(O)-K Nle= norleucine, Met (O)= methionine sulfoxide 1513 GFLSILKKVLPKV-Nle-AH-Met-K Nle= norleucine 1514 GFLSIVKKVLPKV-Nle-AH-Met(O)-K Nle= norleucine, Met (O)= methionine sulfoxide 1515 GFLSIVKKVLPKV-Nle-AH-Met-K Nle= norleucine 1649 KWKKLLKKaLKLLKKLLK a=Nala (Ala-peptoid) 1650 KWKKLLKKLaKLLKKLLK a=Nala (Ala-peptoid) 1651 KWKKLLKKLLaLLKKLLK a=Nala (Ala-peptoid) 1652 KWKKLLaKLLaLLKKLLK a=Nala (Ala-peptoid) 1654 KWKKLLKKaLKLLKKLLK a=Nala (Ala-peptoid) 1655 KWKKLLKKLaKLLKKLLK a=Nala (Ala-peptoid) 1656 KWKKLLKKLLaLLKKLLK a=Nala (Ala-peptoid) 1657 KWKKLLaKLLaLLKKLLK a=Nala (Ala-peptoid) 1737 GKGLTicOicGRTicOicGFTicOicGRTicOicGFTicOicGRTicOicGKR Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1738 GKGLTicOicGRTicOicGFTicOicGRTicOicGFTicOicGRTicOicGKR Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1739 GKGLTicOicGLTicOicGKTicOicGLTicOicGKTicOicGLTicOicGLR Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1740 GKGLTicOicGLTicOicGKTicOicGLTicOicGKTicOicGLTicOicGLR Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1741 GKGLTicOicGKTicOicGLTicOicGKTicOicGLTicOicGKTicOicGKR Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1742 GKGLTicOicGKTicOicGLTicOicGKTicOicGLTicOicGKTicOicGKR Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1743 GKGLTicOicFKTicOicKFTicOicFKTicOicKFTicOicFKTicOicFKR Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1744 GKGLTicOicFKTicOicKFTicOicFKTicOicKFTicOicFKTicOicFKR Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1745 GKGLTicOicGRTicOicGFTicOicGRTicOicGFTicOicELMNS Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1746 GKGLTicOicGRTicOicGFTicOicGRTicOicGFTicOicELMNS Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1747 ELMNSTicOicGLTicOicGKTicOicGLTicOicGKTicOicELMNS Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1748 ELMNSTicOicGLTicOicGKTicOicGLTicOicGKTicOicELMNS Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1749 ELMNSTicOicGKLGKTicOicELMS Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1750 ELMNSTicOicGKLGKTicOicELMS Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1751 ELSTicOicGKGTicOicLKES Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1752 ELSTicOicGKGTicOicLKES Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1753 GKGLTicOicβAlaKTicOicβAlaFTicOicβAlaKTicOicβAlaFTicOicELMNS Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid, βAla- β-alanine 1754 GKGLTicOicβAlaKTicOicβAlaFTicOicβAlaKTicOicβAlaFTicOicELMNS Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid, βAla- β-alanine 1755 EGKGLGβAlaβAlaKTicOicβAlaFTicOicβAlaETicOicβAlaFTicOicELMNS Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid, βAla- β-alanine 1756 EGKGLGβAlaβAlaKTicOicβAlaFTicOicβAlaETicOicβAlaFTicOicELMNS Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid, βAla- β-alanine 1757 KLTicOicKTicOicFTicOicKTicOicFTicOicKTicOicKR Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1758 KLTicOicKTicOicFTicOicKTicOicFTicOicKTicOicKR Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1759 GFTicOicGKTicOicGFTicOicGKTicKKKK Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1760 GFTicOicGKTicOicGFTicOicGKTicKKKK Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1761 GFTicOicGKTicOicGFTicOicGKTicKKKK Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1762 GFTicOicGKTicOicGFTicOicGKTicKKKK Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1763 KLTicOicGKTicOicGFTicOicGKTicKKKK Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1764 KLTicOicGKTicOicGFTicOicGKTicKKKK Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1765 FTicOicKTicOicFTicOicKTicKKKK Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1766 FTicOicKTicOicFTicOicKTicKKKK Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1767 GABAFTicOicGABAKTicOicGABAFTicOicGABAKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid, GABA= γ-aminobutyric acid 1768 GABAFTicOicGABAKTicOicGABAFTicOicGABAKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid, GABA= γ-aminobutyric acid 1769 GTicOicKTicOicGTicOicKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1770 GTicOicKTicOicGTicOicKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1771 GFOicGKOicGFOicGKKKKK Oic= octahydroindolecarboxylic acid 1772 GFOicGKOicGFOicGKKKKK Oic= octahydroindolecarboxylic acid 1773 GFTicGKTicGFTicGKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid 1774 GFTicGKTicGFTicGKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid 1775 GFTicGGKTicGGFTicGGKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid 1776 GFTicGGKTicGGFTicGGKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid 1777 GFG-Oic-GKG-Oic-GFG-Oic-GKGKKKK Oic= octahydroindolecarboxylic acid 1778 GFGOicGKGOicGFGOicGKGKKKK Oic= octahydroindolecarboxylic acid 1779 GFFOicGKFOicGFFOicGKFKKKK Oic= octahydroindolecarboxylic acid 1780 GFFOicGKFOicGFFOicGKFKKKK Oic= octahydroindolecarboxylic acid 1781 βAlaFTicOicβAlaKTicOicβAlaFTicOicβAlaKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid, βAla- β-alanine 1782 βAlaFTicOicβAlaKTicOicβAlaFTicOicβAlaKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid, βAla- β-alanine 1783 AhxFTicOicAhxKTicOicAhxFTicOicAhxKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid, Ahx= 6-aminohexanoic acid 1784 AhxFTicOicAhxKTicOicAhxFTicOicAhxKTicKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid, Ahx= 6-aminohexanoic acid 1785 FTicOicKTicOicFTicOicKTicKKKKKK Tic- tetrahydroisoquinolinecarboxylic acid, Oic- octahydroindolecarboxylic acid 1786 FTicOicKTicOicFTicOicKTicKKKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1787 GFTicOicGKTicOicGFTicOicGKTicKKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1788 GFTicOicGKTicOicGFTicOicGKTicKKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid 1789 GABAFTicOicGABAKTicOicGABAFTicOicGABAKTicKKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid, GABA= γ-aminobutyric acid, 1790 GABAFTicOicGABAKTicOicGABAFTicOicGABAKTicKKKKK Tic= tetrahydroisoquinolinecarboxylic acid, Oic= octahydroindolecarboxylic acid, GABA= γ-aminobutyric acid, 1810 HFLLTLVN-Chg-AKKIL Chg: cyclohexylglycine 1811 HFLLTLVNLAKK-Chg-L Chg: cyclohexylglycine 1812 HFLLTLVN-Chg-AKK-Chg-L Chg: cyclohexylglycine 1917 OOWW O= Orinithine 1918 OOWW O= Orinithine 1919 OOWW O= Orinithine 1920 OOWW O= Orinithine 1921 OOWW O= Orinithine 1922 OOWW O= Orinithine 1923 OOFF O= Orinithine 2135 G-Nle-Nle-Orn-Orn-Nle-Aib-Orn-Orn-Aib-Orn-Orn-Aib-Nle-Orn-Orn-Nle-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2136 G-Nle-Nle-Orn-Orn-Nle-Aib-Orn-Orn-Aib-Orn-Orn-Aib-Nle-Orn-Orn-Nle-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2137 G-Orn-Orn-Nle-Aib-Orn-Orn-Aib-Orn-Orn-Aib-Nle-Orn-Orn-Nle-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2138 G-Orn-Orn-Nle-Aib-Orn-Orn-Aib-Orn-Orn-Aib-Nle-Orn-Orn-Nle-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2139 G-Nle-Aib-Orn-Orn-Aib-Orn-Orn-Aib-Nle-Orn-Orn-Nle-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2140 G-Nle-Aib-Orn-Orn-Aib-Orn-Orn-Aib-Nle-Orn-Orn-Nle-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2141 G-Nle-Aib-Orn-Orn-Nle-Aib-Orn-Orn-Aib-Orn-Orn-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2142 G-Nle-Aib-Orn-Orn-Nle-Aib-Orn-Orn-Aib-Orn-Orn-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2143 G-Orn-Orn-Aib-Orn-Orn-Aib-Nle-Orn-Orn-Nle-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2144 G-Orn-Orn-Aib-Orn-Orn-Aib-Nle-Orn-Orn-Nle-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2145 G-Nle-Aib-Orn-Orn-Aib-Aib-Orn-Orn-Nle-Nle-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2146 G-Nle-Aib-Orn-Orn-Nle-Aib-Orn-Orn-Nle-Nle-Orn-GY Aib= α-aminoisobutyric acid, Nle= norleucine, Orn= ornithine 2148 FLPLLAGLAANFLPKIFC-Acm-KITRKC-Acm Acm= acetamidomethyl 2150 FLPLLAGLC-Acm-KITRKC-Acm-AANFLPKIF Acm=acetamidomethyl 2281 FFHLHFH-dcΔDOPA dcΔDOPA=decarboxy-(E)α,β-dehydro3,4-dihydroxyphenylalanine 2282 FFHLHFH-dcΔDOPA dcΔDOPA=decarboxy-(E)α,β-dehydro3,4-dihydroxyphenylalanine 2622 QC*RRLCYKQRCVTYC*RGR C*: Cystein is protected by Acm 2675 KIGAK-L-CF3-Bpg-KIGAKIKIGAKI CF3-Bpg ie [3-(trifluoromethyl)-bicyclopent-[1.1.1]-1-ylglycine] 2676 KIGAK-L-CF3-Bpg-KIGAKIKIGAKI CF3-Bpg ie [3-(trifluoromethyl)-bicyclopent-[1.1.1]-1-ylglycine] 2679 KIGAKIK-L-CF3-Bpg-GAKIKIGAKI CF3-Bpg ie [3-(trifluoromethyl)-bicyclopent-[1.1.1]-1-ylglycine] 2680 KIGAKIK-L-CF3-Bpg-GAKIKIGAKI CF3-Bpg ie [3-(trifluoromethyl)-bicyclopent-[1.1.1]-1-ylglycine] 2683 KIGAKIKIGAK-L-CF3-Bpg-KIGAKI CF3-Bpg ie [3-(trifluoromethyl)-bicyclopent-[1.1.1]-1-ylglycine] 2684 KIGAKIKIGAK-L-CF3-Bpg-KIGAKI CF3-Bpg ie [3-(trifluoromethyl)-bicyclopent-[1.1.1]-1-ylglycine] 2687 KIGAKIKIGAKIK-L-CF3-Bpg-GAKI CF3-Bpg ie [3-(trifluoromethyl)-bicyclopent-[1.1.1]-1-ylglycine] 2688 KIGAKIKIGAKIK-L-CF3-Bpg-GAKI CF3-Bpg ie [3-(trifluoromethyl)-bicyclopent-[1.1.1]-1-ylglycine] 2714 GWLDVAKKIGKAAFNVAKNFL-spacer-LFNKAVNFAAKGIKKAVDLWG Spacer = 8-amino-octanoic acid 2715 GWLDVAKKIGKAAFNVAKNFL-spacer-LFNKAVNFAAKGIKKAVDLWG Spacer = 8-amino-3,6-dioxaoctanoic acid 2747 GFLSILKKVLPKVXAHXK X; Nle 2748 GFLSILKKVLPKSXAHSK X; Nle 2749 GFLSSLKKSLPKVXAHXK X; Nle 2750 GFLSSLKKSLPKSXAHSK X; Nle 2751 GFRSILKKVSPKVXAHXK X; Nle 2752 GFRSILKKVSPKVXAHXK X; Nle 2753 GFLSSLKKSLGKSXAHSK X; Nle 2754 GFLSSLKKSLAKSXAHSK X; Nle 2840 FVQWFSKFLGOIL Ornithine 2973 GRPNPVNNKPT*PHPRL *=α-GalNAc 2975 GKPRPYSPRPT*SHPRPIRV *=α-GalNAc 3027 I*LPWKWPWWPWRR *=Reduced amide bond ψ[CH2NH] 3028 ILPWKWPW*WPWRR *=Reduced amide bond ψ[CH2NH] 3029 I*LPWKWPW*WPWRR *=Reduced amide bond ψ[CH2NH] 3031 I*LPWKWPWWPWRR *=Reduced amide bond ψ[CH2NH] 3032 ILPWKWPW*WPWRR *=Reduced amide bond ψ[CH2NH] 3033 I*LPWKWPW*WPWRR *=Reduced amide bond ψ[CH2NH] 3035 I*LPWKWPWWPWRR *=Reduced amide bond ψ[CH2NH] 3036 ILPWKWPW*WPWRR *=Reduced amide bond ψ[CH2NH] 3037 I*LPWKWPW*WPWRR *=Reduced amide bond ψ[CH2NH] 3039 I*LPWKWPWWPWRR *=Reduced amide bond ψ[CH2NH] 3040 ILPWKWPW*WPWRR *=Reduced amide bond ψ[CH2NH] 3041 I*LPWKWPW*WPWRR *=Reduced amide bond ψ[CH2NH] 3085 GLKKIFKAGLGSLVKGIK*AHVAS *=palmitate(PAL) 3145 VDIHVWD*GV D*=β-aspartic acid 3565 XALWKNMLKGIGKLAGKAALGAVKKLVGAES X=H 3566 XALWMTLLKKVLKAAAKAALNAVLVGANA X=H 3570 KKALLOHALHOLALLAOHLAHOLKKA O=Ornithine 3571 ALALLOHALHOLALLAOHLAHOLALA O=Ornithine 3572 FFKKLOHALHOLALLAOHLAHOLKKA O=Ornithine 3573 KKALLOHPLHOLALLAOHLAHOLKKA O=Ornithine 3732 LNWGA-Abu-LKH-Abu-Abu-K Abu 2 =aminobutyric acid 3737 LNWGA-Nle-LKH-Nle-Nle-K Nle =norleucine 3738 LNWGA-Aca-LKH-Aca-Aca-K Aca 1 =aminocyclohexane carboxylic acid 3741 LDVKKII-Abu-VA-Abu-KIKPNPA-Abu-KKI-Abu-PK Abu 2 =aminobutyric acid 3743 LDVKKII-Abu-VA-Abu-KIRPNPA-Abu-KKI-Abu-PK Abu 2 =aminobutyric acid 3808 Aib-P-Aib-A-Aib-AQ-Aib-V-Aib-GL-Aib-PV-Aib-Aib-EQ Aib = α- methylalanine 3913 INWLKLGKK-Nle-Nle-SAL Nle 3948 IL-(Nlys)-WKW-(Nlys)-WW-(Nlys)-WRR Nlys 3967 VRRF-(Nphe)-WWW-(Nphe)-FLRR Nphe 3968 VRRF-(Nlys)-WWW-(Nlys)-FLRR Nlys 3970 VRRF-(Nleu)-WWW-(Nleu)-FLRR Nleu 3972 KKF-(Nlys)-WWW-(Nlys)-FKK Nlys 3984 KWKLFKKI-Nala-KFLHLAKKF Nala 4194 ZCRRLCYKQRCVTYCRGR Z= pyroglutamic acid 4195 ZSRRLSYKQRSVTYSRGR Z= pyroglutamic acid 4196 ZSRRLCYKQRCVTYSRGR Z= pyroglutamic acid 4197 ZCRRLSYKQRSVTYCRGR Z= pyroglutamic acid 4198 ZDRRLSYKQRSVTYORGR Z= pyroglutamic acid 4199 ZSRRLDYKQROVTYSRGR Z= pyroglutamic acid 4200 ZCRRLEYKQRKVTYCRGR Z= pyroglutamic acid 4201 ZERRLCYKQRCVTYKRGR Z= pyroglutamic acid