SMDBid | siRNA (sense/antisense) 5'>3' | Modification (sense/antisense) | Position (sense/antisense) |
Modified component (sense/antisense) |
Efficacy (%) | Reference |
SM0022 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGC |
2-Aminoethyl 2-O-Methyl |
5,19,20 2 |
Sugar Sugar |
45.9 percent target mRNA inhibition | 19282453 |
SM0025 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGC |
4-C-Hydroxymethyl Deoxyribonucleic acid 2-O-Methyl |
5,19,20 2 |
Sugar Sugar |
74.6 percent target mRNA inhibition | 19282453 |
SM0068 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGCU |
2-Aminoethyl 2-O-Methyl* 2-Aminoethyl |
5,19,20 1 * 21 |
Sugar Sugar |
71 percent target mRNA inhibition | 19282453 |
SM0071 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGCU |
4-C-Hydroxymethyl Deoxyribonucleic acid 2-O-Methyl* 2-Aminoethyl |
5,19,20 1 * 21 |
Sugar Sugar |
88 percent target mRNA inhibition | 19282453 |
SM0113 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGCU |
2-Aminoethyl 2-O-Methyl* 2-Cyanoethyl |
5,19,20 1 * 18 |
Sugar Sugar |
37.7 percent target mRNA inhibition | 19282453 |
SM0116 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGCU |
4-C-Hydroxymethyl Deoxyribonucleic acid 2-O-Methyl* 2-Cyanoethyl |
5,19,20 1 * 18 |
Sugar Sugar |
45.5 percent target mRNA inhibition | 19282453 |
SM0158 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGC |
2-Aminoethyl Altritol nucleic acid |
5,19,20 1,2 |
Sugar Sugar |
39.4 percent target mRNA inhibition | 19282453 |
SM0161 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGC |
4-C-Hydroxymethyl Deoxyribonucleic acid Altritol nucleic acid |
5,19,20 1,2 |
Sugar Sugar |
57.5 percent target mRNA inhibition | 19282453 |
SM0203 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGCU |
2-Aminoethyl Altritol nucleic acid |
5,19,20 20,21 |
Sugar Sugar |
87.3 percent target mRNA inhibition | 19282453 |
SM0206 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGCU |
4-C-Hydroxymethyl Deoxyribonucleic acid Altritol nucleic acid |
5,19,20 20,21 |
Sugar Sugar |
92.2 percent target mRNA inhibition | 19282453 |
SM0248 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGCU |
2-Aminoethyl Altritol nucleic acid |
5,19,20 5,8,11,14,17,20 |
Sugar Sugar |
9.9 percent target mRNA inhibition | 19282453 |
SM0251 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGCU |
4-C-Hydroxymethyl Deoxyribonucleic acid Altritol nucleic acid |
5,19,20 5,8,11,14,17,20 |
Sugar Sugar |
25.2 percent target mRNA inhibition | 19282453 |
SM0293 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGCU |
2-Aminoethyl Altritol nucleic acid |
5,19,20 3,6,14,18,20,21 |
Sugar Sugar |
46.6 percent target mRNA inhibition | 19282453 |
SM0296 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGCU |
4-C-Hydroxymethyl Deoxyribonucleic acid Altritol nucleic acid |
5,19,20 3,6,14,18,20,21 |
Sugar Sugar |
76.5 percent target mRNA inhibition | 19282453 |
SM0338 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGT |
2-Aminoethyl Hexitol nucleic acid* 2-Deoxy |
5,19,20 18,19,20 * 21 |
Sugar Sugar |
83.4 percent target mRNA inhibition | 19282453 |
SM0341 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGT |
4-C-Hydroxymethyl Deoxyribonucleic acid Hexitol nucleic acid* 2-Deoxy |
5,19,20 18,19,20 * 21 |
Sugar Sugar |
84.8 percent target mRNA inhibition | 19282453 |
SM0383 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGT |
2-Aminoethyl Hexitol nucleic acid* 2-Deoxy |
5,19,20 2,18,19,20 * 21 |
Sugar Sugar |
72 percent target mRNA inhibition | 19282453 |
SM0386 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGT |
4-C-Hydroxymethyl Deoxyribonucleic acid Hexitol nucleic acid* 2-Deoxy |
5,19,20 2,18,19,20 * 21 |
Sugar Sugar |
84.4 percent target mRNA inhibition | 19282453 |
SM0428 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGT |
2-Aminoethyl Hexitol nucleic acid* 2-Deoxy |
5,19,20 3,18,19,20 * 21 |
Sugar Sugar |
73.2 percent target mRNA inhibition | 19282453 |
SM0431 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGT |
4-C-Hydroxymethyl Deoxyribonucleic acid Hexitol nucleic acid* 2-Deoxy |
5,19,20 3,18,19,20 * 21 |
Sugar Sugar |
85.7 percent target mRNA inhibition | 19282453 |
SM0473 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGT |
2-Aminoethyl Hexitol nucleic acid* 2-Deoxy |
5,19,20 2,9,18,19,20 * 21 |
Sugar Sugar |
11.7 percent target mRNA inhibition | 19282453 |
SM0476 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGT |
4-C-Hydroxymethyl Deoxyribonucleic acid Hexitol nucleic acid* 2-Deoxy |
5,19,20 2,9,18,19,20 * 21 |
Sugar Sugar |
19.7 percent target mRNA inhibition | 19282453 |
SM0518 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGT |
2-Aminoethyl 2-Aminoethoxymethyl* 2-Deoxy |
5,19,20 18,19 * 21 |
Sugar Sugar |
30 percent target mRNA inhibition | 19282453 |
SM0521 |
GACGTAAACGGCCACAAGTTC ACUUGUGGCCGUUUACGUCGT |
4-C-Hydroxymethyl Deoxyribonucleic acid 2-Aminoethoxymethyl* 2-Deoxy |
5,19,20 18,19 * 21 |
Sugar Sugar |
51.8 percent target mRNA inhibition | 19282453 |
SM0563 |
GACGUAAACGGCCACAAGUUC ACUUGUGGCCGUUUACGUCGT |
2-Aminoethyl 2-Aminopropoxymethyl* 2-Deoxy |
5,19,20 18,19 * 21 |
Sugar Sugar |
16.1 percent target mRNA inhibition | 19282453 |