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IDPMIDSEQUENCENAME LENGTHACTIVITY
103314499271FLPLLAGLAANFLPTIICKISYKCGGN624IC50=4.88 µg/ml
103414499271LLAGLAANFLPTIICKISYKCPTP121IC50=>100 µg/ml
103514499271FAGLAANFLPTIICKISYKCPTP220IC50=>100 µg/ml
103614499271FLKLLKKLAAKFLPTIICKISYKCPTP424IC50=18.1 µg/ml
103714499271FLKLLKKLAAKLFPTP513IC50=5.43 µg/ml
103814499271FLKLLKKLAAKLFPTP613IC50=17.56 µg/ml
103914499271FLGALFKALSKLLPTP713IC50=5.25 µg/ml
104014499271FLKLLAGLLKNFAPTP813IC50=32.23 µg/ml
105918617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=15.1 µg/ml
106018617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=11.5 µg/ml
106118617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=11.3 µg/ml
106218617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=11.7 µg/ml
106318617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=11.3 µg/ml
106418617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=10.6 µg/ml
106518617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=12.9 µg/ml
106618617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=23.9 µg/ml
111912005420KWKLFKKIPKFLHSAKKFCA-MA-P18IC50=20 µM
112012005420KWKFKKIPKFLHLAKKFP1817IC50=8 µM
112112005420KWKLFKKILKFLHLAKKF[L9]-P1818IC50=3 µM
112212005420KWKLFKKISKFLHLAKKF[S9]-P1818IC50=4 µM
112312005420WKLFKKIPKFLHLAKKFN-117IC50=9.5 µM
112412005420FKLFKKIPKFLHLAKKFN-217IC50=11 µM
112512005420KWFKKIPKFLHLAKKFN-316IC50=17 µM
112612005420WFKKIPKFLHLAKKFN-415IC50=32 µM
112712005420WKKIPKFLHLAKKFN-514IC50=100. <µM
112812005420WFKKIPKFLHLLKKFN-3L15IC50=5 µM
112912005420WKKIPKFLHLLKKFN-4L14IC50=5 µM
113012005420WKKIPKFLHLLKKFN-5L14IC50=17 µM
113112005420KWKLFKKIPFLHLAKKFC-117IC50=26 µM
113212005420KWKLFKKIPKFLHLAKKC-217IC50=38 µM
113312005420KWKLFKKIPLHLAKKFC-316IC50=79 µM
113412005420KWKLFKKIPKFLHLAKC-416IC50=54 µM
113512005420KWKLFKKIPHLAKKFC-515IC50=100 µM
113612005420KWKLFKKIPKFLHLAC-615IC50=47 µM
113712005420KWKLFKKIPLAKKFC-714IC50=100. <µM
113812005420KWKLFKKIPKFLHLC-814IC50=83 µM
113912005420KWKLFKKIPLKKFC-913IC50=100. <µM
114012005420KWKLFKKIPKFLHC-1013IC50=100. <µM
119710675500KWKLFKKIGIGKFLHSAKKFCA-MA20IC50=44 µM
119810675500KWKLFKKIKFLHSAKKFCA-MA117IC50=100 µM
119910675500KWKLFKKIPKFLHSAKKFCA-MA218IC50=28 µM
120010675500KWKLFKKIGPGKFLHSAKKFCA-MA320IC50=>100 µM
12327849420KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKALCecropin B35IC50=24.8 µM
12367849420SWLSKTAKKLENSAKKRISEGIAIAIQGGPRCecropin P131IC50=>100 µM
12407849420MPRWRLFRRIDRVGKQIKQGILRAGPAIALVGDARAVGShiva-138IC50=56 µM
12487849420KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKALCecropin B35IC50=42.5 µM
12517849420KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKALCecropin B35IC50=24.5
125210951191GLFDIIKKIAESFAurein1.213LC50 = 10 µM
126110951191GLFDIVKKVVGAFGSLAurein2.516LC50 = 10 µM
127010951191GLFDIAKKVIGVIGSLAurein2.616LC50 = 10 µM
127910951191GLFDIVKKIAGHIAGSIAurein 3.117LC50=10-100 µM
128810951191GLFDIVKKIAGHIASSIAurein 3.217LC50 = 10 µM
129710951191GLFDIVKKIAGHIVSSIAurein 3.317LC50 = 10 µM
14021708887, 2285300GIGKFLHAAKKFAKAFVAEIMNSMagainin B23IC50=37 µg/ml
14031708887, 2285300GIGKFLHSAKKFAKAFVAEIMNSMagainin G23IC50=42 µg/ml
14041708887, 2285300AIGKFLHSAKKFGKAFVGEIMNSMagainin A23IC50=49 µg/ml
14051708887, 2285300ALSKALSKALSKALSKALSKALSKZ4424Not Available
14061708887, 2285300ALSKALSKALSKALSKALSKALSKZ2424Not Available
14071708887, 2285300GIGKFLHSAKKFGKAFVGEIMNSMagainin 223IC50 >200 µg/ml
146521252288KWKSFAKTFKSAKKTVAHTALKAISSL6A/L17A26IC50=>83.6 µMo/L
146621252288KWKSFLKTFKSAKKTVAHTAAKAISSL17A/L21A26IC50=>83.6 µMo/L
146721252288KWKSFLKTFKSAKKTVAHTALKAISSL17A26IC50=>83.6 µMo/L
146821252288KWKSFLKTFKSAKKTVAHTAAKAISSL21A26IC50=70.8 µMo/L
146921252288KWKSFAKTFKSAKKTVLHTALKAISSL6A26IC50=62.3 µMo/L
147021252288KWKSFLKTFKSAKKTVLHTALKAISSP26IC50=15.8 µMo/L
147121252288KWKSFLKTFKSLKKTVLHTALKAISSA12L26IC50=5 µMo/L
147221252288KWKSFLKTFKSAKKTVLHTLLKAISSA20L26IC50=5.1 µMo/L
147321252288KWKSFLKTFKSLKKTVLHTLLKAISSA12L/A20L26IC50=6.2 µMo/L
147421252288KWKSFLKTFKSLKKTVLHTLLKLISSA12L/A20L/A23L26IC50=5.7 µMo/L
161912366526PEWFKCRRWQWRMKKLGAL118IC50=>404 µM
162012366526PAWFKARRWAWRMKKLAAL218IC50=>254 µM
162112366526PAWRKAFRWAWRMKKLAAL318IC50=18 µM
162212366526PAWFKARRWAWRMLKKAAL418IC50=16 µM
162312366526PAWRKAFRWAWRMLKKAAL518IC50=8 µM
162412366526PAWRKAFRWAARMLKKAAL618IC50=12 µM
162512366526PAWRKAFRAAWRMLKKAAL718IC50=11 µM
162612366526PAWAKAFRAAARMKLKAAL818IC50=87 µM
162712366526PAWRKAARWAWRMLKKAAL918IC50=32 µM
162812366526PAARKAFRWAWRMLKKAAL1018IC50=20 µM
162912366526PAARKAARWAWRMLKKGAL1118IC50=75 µM
163012366526PAWRKAFRWAKRMLKKAAL1218IC50=10 µM
163112366526PAWRKAFRKAWRMLKKAAL1318IC50=12 µM
163212366526PAWRKARRWAWRMKKLAAL1418IC50=141 µM
163312366526PAWRKARRWARRMKKLAAL1518IC50=92 µM
170222641352LLRHVVKILEKYLTemporin-La1324.15Inhibition ratio at 50 µg/ml
170322641352LLRHVVKILSKYLTemporin-Las1327.99 Inhibition ratio at 50 µg/ml
170422641352RGDLLRHVVKILEKYLRGD-La1619.76 Inhibition ratio at 50 µg/ml
170522641352RGDLLRHVVKILSKYLRGD-Las1629.33 Inhibition ratio at 50 µg/ml
17069614066ALWKNMLKGIGKLAGQAALGAVKTLVGADRS B328Cytotoxicity =12 µM
17079614066ALWKDILKNVGKAAGKAVLNTVTDMVNQDRS B428Cytotoxicity =15 µM
17089614066ALWKTMLKKLGTMALHAGKAALGAAADTISQGTQDRS S135Not Available
1773NoneFALALKALKKALKKLKKALKKALHecate Ac23LD50 =54 µg/ml
1774NoneFALALKALKKALKKLKKALKKALHecate AM23LD50 =23 µg/ml
1775NoneMPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALGSB-37 AC38LD50 =175 µg/ml
1776NoneMPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALGSB-37 AM38LD50 =540 µg/ml
1777NoneFAKKLAKKLKKLAKKLAKLALALSHIVA 10 AC23LD50 =>1000 µg/ml
1778NoneFALAAKALKKLAKKLKKLAKKALFLAK01 AM23LD50 =62 µg/ml
1779NoneFALALKALKKLLKKLKKLAKKALFLAK03 AM23LD50 =26 µg/ml
1780NoneFALALKALKKLAKKLKKLAKKALFLAK04 AM23LD50 =10 µg/ml
1781NoneFALAKLAKKAKAKLKKALKALFLAK05 AM21LD50 =74 µg/ml
1782NoneFALALKALKKLKKALKKALFLAK06 AM19LD50 =14 µg/ml
1783NoneFALALKALKKLKKALKKALFLAK06 AC19LD50 =65 µg/ml
1784NoneFAKKLAKKLKKLAKLALALFLAK06 R-AC19LD50 =140 µg/ml
1785NoneVALALKALKKALKKLKKALKKALKAL V23LD50 =72 µg/ml
1786NoneFALALKKALKALKKALFLAK 17 AM16LD50 =21 µg/ml
1787NoneFAKKLAKLAKKLAKLALFLAK 26 AM17LD50 =9 µg/ml
1788NoneFAKKLAKLAKKLAKLALALFLAK 25 AM19LD50 =9 µg/ml
1789NoneFALALKALKKALkkLKKALKKALHECATE 2DAc23LD50 =14 µg/ml
1790NoneFAKKLAKLAKKLLALFLAK43 AM15LD50 =17 µg/ml
1791NoneFAKKLAKLAKKALALFLAK44 AM15LD50 =130 µg/ml
1792NoneFALAKKALKKAKKALFLAK62 AM15LD50 =760 µg/ml
1793NoneFAKKLAKKLKKLAKLALAKFLAK 06R-AM19LD50 =98 µg/ml
1794NoneGIGKFLKKAKKFGKAFVKILKKMSI-78 AM22LD50 =31 µg/ml
1795NoneFAKLLAKLAKKLLFLAK5013LD50 =9 µg/ml
1796NoneFAKKLAKLALKLAKLFLAK5115LD50 =140 µg/ml
1797NoneFAKKLAKKLAKLALFLAK5714LD50 =260 µg/ml
1798NoneFAKKLKKLAKLAKKLFLAK7115LD50 =300 µg/ml
1799NoneFAKKALKALKKLFLAK7712LD50 =575 µg/ml
1800NoneVAKLLAKLAKKLLFLAK50V13LD50 =23 µg/ml
1801NoneFAKLLAKLAKKLFLAK50F12LD50 =40 µg/ml
1802NoneVAKKLAKLAKKLAKLALFLAK26V AM17LD50 =32 µg/ml
1803NoneKWKLFKKIGAVLKVLCAME-1515LD50 =45 µg/ml
1804NoneFAKLLAKLAKKALFLAK50C13LD50 =60 µg/ml
1805NoneFAKLLAKALKKLLFLAK50D13LD50 =16 µg/ml
1806NoneFAKLLKLAAKKLLFLAK 50E13LD50 =500 µg/ml
1807NoneFAKLLAKKLLFLAK8010LD50 =>1000 µg/ml
1808NoneFAKKLAKALLFLAK8110LD50 =>1000 µg/ml
1809NoneFAKKLAKKLLFLAK8210LD50 =31 µg/ml
1810NoneFAKLAKKLLFLAK83M9LD50 =>1000 µg/ml
1811NoneFAKKLAKLAKKLAKLALFLAK 26 Ac17LD50 =105 µg/ml
1812NoneILPWKWPWWPWRRIndolicidin13LD50 =64 µg/ml
1813NoneFAKALKALLKALKALFLAK 17 C15LD50 =80 µg/ml
1814NoneFAKLLAKLAKAKLFLAK 50H13LD50 =475 µg/ml
1815NoneFAKLLAKLAKLKLFLAK 50G13LD50 =90 µg/ml
1816NoneFAKKLAKKLKKLAKKLAKKWKLSHIVA DERIV P69 + KWKL22LD50 =44 µg/ml
1817NoneFAKKLAKKLKKLAKKLAKShiva 10(1-18 AC)18LD50 =190 µg/ml
1818NoneFAKKLAKKLKKLAKKLAKKWKLSHIVA 10 PEPTIDE 71 + KWKL22LD50 =93 µg/ml
1819NoneKWKLFKKKTKLFKKFAKKLAKKLCA (1-7) Shiva10 (1-16)23LD50 =150 µg/ml
1820NoneFAKKLAKKLAKALFLAK 5413LD50 =465 µg/ml
1821NoneFAKKLAKKLAKLLFLAK 5613LD50 =42 µg/ml
1822NoneFAKKLAKKLAKAALFLAK 5814LD50 =970 µg/ml
1823NoneFAKKLAKKAKLAKKLFLAK 7215LD50 =>1000 µg/ml
1824NoneFAKKLKKLAKKLFLAK 7512LD50 =540 µg/ml
1825NoneKTKLFKKFAKKLAKKLKKLAKKLSHIVA 10 (1-16) Ac23LD50 =29 µg/ml
1826NoneKWKLFKKKTKLFKKFAKKLAKKLCA(1-7) Shiva10(1-16)-COOH23LD50 =63 µg/ml
1827NoneILPWKWPWWPWRRIndolocidin-ac13LD50 =12 µg/ml
1828NoneFAKALAKLAKKLLFLAK50B13LD50 =23 µg/ml
1829NoneFAKLLALALKLKLFLAK50I13LD50 =65 µg/ml
1830NoneFAKLLAKLAKAKAFLAK50K13LD50 =>1000 µg/ml
1831NoneFAKLLAKLAKAKGFLAK50L13LD50 =>1000 µg/ml
1832NoneFAKKLAKKLKKLAKKLAKLALALKALALKALShiva-1131LD50 =96 µg/ml
1833NoneFAKKLAKKLKKLAKKLIGAVLKVSHIVA 11[(1-16)ME(2-9]-COOH23LD50 =95 µg/ml
1834NoneFAKLLAKALKLKLFLAK 50N13LD50 =250 µg/ml
1835NoneFAKLLAKALKKALFLAK 50O13LD50 =60 µg/ml
1836NoneFAKLLAKALKKLFLAK 50P12LD50 =46 µg/ml
1837NoneKWKLFKKALKKLKKALKKALCA(1-& HECATE(11/23)20LD50 =11 µg/ml
1838NoneKIAKVALAKLGIGAVLKVLTTGLPYL-ME23LD50 =635 µg/ml
1839NoneFAKKLAKLAKKLFLAG26-D112LD50 =620 µg/ml
1840NoneMPKEKVFLKIEKMGRNIRNVISHNU319LD50 =>1000 µg/ml
1841NoneGIGAVLKVLTTGLPALISWIKRKRQQMELITTIIN26LD50 =9 µg/ml
1842NoneFAKKLAKLAKKLAKALFLAK26-D216LD50 =>1000 µg/ml
1843NoneFAKKLLAKALKLFLAG26-D312LD50 =180 µg/ml
1844NoneFAKFLAKFLKKALFLAK50 Q113LD50 =35 µg/ml
1845NoneFAKLLFKALKKALFLAK50 Q213LD50 =500 µg/ml
1846NoneFAKLLAKFLKKALFLAK50 Q313LD50 =150 µg/ml
1847NoneFAKLLAKAFKKALFLAK50 Q413LD50 =730 µg/ml
1848NoneFAKLFAKAFKKALFLAK50 Q513LD50 =>1000 µg/ml
1849NoneFAKLLAKALKKFLFLAK50 Q613LD50 =70 µg/ml
1850NoneFAKLLAKALKKFALFLAK50 Q714LD50 =54 µg/ml
1851NoneFAKLLAKLAKKFALFLAK50 Q814LD50 =730 µg/ml
1852NoneFAKLFAKLAKKFALFLAK50 Q914LD50 =400 µg/ml
1853NoneFKLAFKLAKKAFLFLAK50 Q1013LD50 =360 µg/ml
1854NoneFAKLLAKLAKFLAK50 T110LD50 =615 µg/ml
1855NoneFAKLLAKLAKKVLFLAK50 T213LD50 =18 µg/ml
1856NoneFAKLLAKLAKKILFLAK50 T313LD50 =90 µg/ml
1857NoneFAKLLAKLAKKELFLAK50 T413LD50 =>1000 µg/ml
1858NoneFAKLLAKLAKKSLFLAK50 T513LD50 =440 µg/ml
1859NoneFAKLAFLAK905LD50 =500 µg/ml
1860NoneFAKLFFLAK915LD50 =>1000 µg/ml
1861NoneKAKLFFLAK925LD50 =>1000 µg/ml
1862NoneKWKLFFLAK935LD50 =600 µg/ml
1863NoneFGKGIGKVGKKLLFLAK50 Z113LD50 =>1000 µg/ml
1864NoneFAFGKGIGKVGKKLLFLAK50 Z215LD50 =>1000 µg/ml
1865NoneFAKAIAKIAFGKGIGKVGKKLLFLAK50 Z322LD50 =>1000 µg/ml
1866NoneFAKLWAKLAFGKGIGKVGKKLLFLAK50 Z422LD50 =54 µg/ml
1867NoneFAKLWAKLAKKLFLAK50 Z512LD50 =500 µg/ml
1868NoneFAKGVGKVGKKALFLAK50 Z613LD50 =>1000 µg/ml
1869NoneFAFGKGIGKIGKKGLFLAK50 Z715LD50 =>1000 µg/ml
1870NoneFAKIIAKIAKIAKKILFLAK50 Z816LD50 =625 µg/ml
1871NoneFAFAKIIAKIAKKIIFLAK50 Z915LD50 =>1000 µg/ml
1872NoneFALALKAFLAK947LD50 =430 µg/ml
1873NoneKWKLAKKALALLFLAK93B12LD50 =44 µg/ml
1874NoneFAKIIAKIAKKIFLAK50 Z1012LD50 =>1000 µg/ml
1875NoneFALALKALKKALFLAK9612LD50 =150 µg/ml
1876NoneFALKALKKFLAK978LD50 =>1000 µg/ml
1877NoneKYKKALKKLAKLLFLAK9813LD50 =110 µg/ml
1878NoneFKRLAKIKVLRLAKIKRFKRLA17LD50 =106 µg/ml
1879NoneFAKLAKKALAKLLFLAK91B13LD50 =315 µg/ml
1880NoneKAKLAKKALAKLLFLAK92B13LD50 =>1000 µg/ml
1881NoneKLALKLALKALKAAKLAFLAK9917LD50 =160 µg/ml
1882NoneFAKLLAKLAKKFLAK50T611LD50 =>1000 µg/ml
1883NoneFAKLLAKLAKKGLFLAK50T713LD50 =430 µg/ml
1884NoneFALKALKKLKKALKKALFLAK9517LD50 =64 µg/ml
1885NoneVAKLLAKLAKKVLFLAK50T813LD50 =315 µg/ml
1886NoneYAKLLAKLAKKALFLAK50T913LD50 =>1000 µg/ml
1887NoneKLLKLLLKLYKKLLKLLFLAK100-CO2H17LD50 =135 µg/ml
1888NoneFAVGLRAIKRALKKLRRGVRKVAKDLFAGVL26LD50 =240 µg/ml
1889NoneKLAKKLAKLAKLAKALModelin-516LD50 =61 µg/ml
1890NoneKLAKKLAKLAKLAKALModelin-5-CO2H16LD50 =320 µg/ml
1891NoneFALALKALKKLFLAK1209LD50 =360 µg/ml
1892NoneFALAKALKKALFLAK12111LD50 =>1000 µg/ml
1893NoneFALALKLAKKALFLAK96B12LD50 =230 µg/ml
1894NoneFALLKLFLAK96G6LD50 =630 µg/ml
1895NoneFALALKALKKFLAK96F10LD50 =510 µg/ml
1896NoneFALKALKKALFLAK96C10LD50 =940 µg/ml
1897NoneFALLKALKKALFLAK96D11LD50 =305 µg/ml
1898NoneKFKKLAKKFModelin-8D9LD50 =>1000 µg/ml
1899NoneKFKKLAKKWModelin-8E9LD50 =>1000 µg/ml
1900NoneFALALKALKKAFlak 96H11LD50 =>1000 µg/ml
1901NoneFALLKALLKKALFlak 96I12LD50 =190 µg/ml
1902NoneFALALKLAKKLFlak 96J11LD50 =770 µg/ml
1903NoneLKKLAKLALAFFlak 96L11LD50 =555 µg/ml
1904NoneVALALKALKKLFLAK-120G11LD50 =950 µg/ml
1905NoneFALALKLKKLFLAK-120D10LD50 =550 µg/ml
1906NoneFALALKAKKLFLAK-120C10LD50 =>1000 µg/ml
1907NoneFALAFLAK-120B4LD50 =>1000 µg/ml
1908NoneWALALFLAK-120F5LD50 =260 µg/ml
1909NoneGIGKFLHAAKKFAKAFVAEIMNSMagainin2wisc23LD50 =22 µg/ml
1910NoneFAKKFAKKFKKFAKKFAKFAFAFD2A2123LD50 =64 µg/ml
1911NoneKKVVFKVKFKKSL-110LD50 =340 µg/ml
1912NoneFKVKFKVKVKKSL-710LD50 =315 µg/ml
1913NoneLPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALGLSB-3738LD50 =50 µg/ml
1914NoneFAKKLAKKLKKLAKKLAKLAKKLAnubis-223LD50 =38 µg/ml
1915NoneFAKKLAKLAKKLAKLALALFLAK 17 CV19LD50 =23 µg/ml
1916NoneVAKFLAKFLKKALFLAK50 Q1V13LD50 =92 µg/ml
1917NoneVAKKFAKKFKKFAKKFAKFAFAFD2A21V23LD50 =210 µg/ml
1918NoneVAKKLAKLAKKLAKLALALFLAK 25 AM V19LD50 =130 µg/ml
1919NoneVAKKLAKLAKKLLALFLAK43 AM V15LD50 =86 µg/ml
1920NoneVAKLLAKALKKLLFLAK50D V13LD50 =45 µg/ml
1921NoneVALALKALKKALKKLKKALKKALHecate AM V23LD50 =340 µg/ml
1922NoneVALALKALKKALKKLKKALKKALHecate AC V23LD50 =160 µg/ml
1923NoneVALALKALKKLAKKLKKLAKKALFLAK04 AM V23LD50 =84 µg/ml
1924NoneFAKLLAKLAKKAAFLAK50J13Not Available
281623000474RRRRRNWMWC9R10IC50=39 µM
281723000474RRRRRWCMNW9S1R10IC50=18 µM
281823000474RRRRRNWMWC9R10IC50=29 µM
281923000474RRRRRWCMNW9S1R10IC50=12 µM
282023000474RRRRRNWMWC9R10IC50=16 µM
282123000474RRRRRWCMNW9S1R10IC50=10 µM
284923028527GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAVAdenoregulin33GI50 =8.06±0.50 µM
285123577112, 21871946FVDLKKIANIINSIFTempoprin-1CEa1522% Cell viability at 40 µM
285223577112, 21871946FVDLKKIANIINSIFTempoprin-1CEa1561% Cytotoxicity at 40 µM
285323577112, 21871946FVDLKKIANIINSIFTempoprin-1CEa1561% Cell viability at 40 µM
285423577112, 21871946FVDLKKIANIINSIFTempoprin-1CEa1532% Cytotoxicity at 40 µM
286122084165KLlLKlLkkLLKlLKKKLytik17IC50=18.5 µMol/L
286822084165KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKKIL-4RaÐlytic hybrid peptide33IC50=5.7 µMol/L
287223583573DEVDcaspase 3 inhibitor465% Cell viability at 20 µM
287323583573DEVDcaspase 3 inhibitor440% Cell viability at 30 µM
287423583573DEVDcaspase 3 inhibitor435 % Cell viability at 40 µM
287523583573FVDLKKIANIINSIFTempoprin-1CEa1570% Cell viability at 20 µM
287623583573FVDLKKIANIINSIFTempoprin-1CEa1545% Cell viability at 30 µM
287723583573FVDLKKIANIINSIFTempoprin-1CEa1530 % Cell viability at 40 µM
288020212453KWKLFKKIGAVLKVLCamel15LC50 = 6.2 µM
290121849092KLlLKlLkkLLKlLKKKLytik17IC50= 34.5 µM
290221849092KLlLKlLkkLLKlLKKKLytik17IC50= 14.1 µM
290321849092KLlLKlLkkLLKlLKKKLytik17IC50= 25.7 µM
290421849092KLlLKlLkkLLKlLKKKLytik17IC50= 27.0 µM
290521849092KLlLKlLkkLLKlLKKKLytik17IC50= 20.0 µM
290621849092KLlLKlLkkLLKlLKKKLytik17IC50= 19.4 µM
291321849092THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKKTransferrin receptor (TfR)-lytic hybrid peptide32IC50= 8.8 µM
291421849092THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKKTransferrin receptor (TfR)-lytic hybrid peptide32IC50= 4.0 µM
291521849092THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKKTransferrin receptor (TfR)-lytic hybrid peptide32IC50= 6.5 µM
291621849092THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKKTransferrin receptor (TfR)-lytic hybrid peptide32IC50= 7.8 µM
291721849092THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKKTransferrin receptor (TfR)-lytic hybrid peptide32IC50= 4.8 µM
291821849092THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKKTransferrin receptor (TfR)-lytic hybrid peptide32IC50= 9.3 µM
309616004618MRKEFHNVLSSGQLLADKRPARDYNRKPep2727IC50= >70 µM
309716004618MWKWFHNVLSSWQLLADKRPARDYNRKPep27anal127IC50= 55 µM
309816004618MWKWFHNVLSWWWLLADKRPARDYNRKPep27anal227IC50= <10 µM
309916004618MRKWFHNVLSSGQLLADKWPAWDYNRKPep27anal327IC50= 38 µM
310016004618MWKEFHNVLSSGQLLADKRWARWYNRWPep27anal427IC50= 29 µM
310116004618MWKWFHNVLSSGQLLADKWWAWWYNWWPep27anal527IC50=>70 µM
311423993331KWLRRVWRWWRMAP-04-0311Cell viability >80% at 25 µM
311523993331KWLRRVWRWWRMAP-04-0311Cell viability ~50% at 50 µM
311623993331KWLRRVWRWWRMAP-04-0311Cell viability <40% at 75 µM
311723993331KWLRRVWRWWRMAP-04-0311Cell viability >20% at 100 µM
311823993331KWLRRVWRWWRMAP-04-0311Cell viability ~100% at 25 µM
311923993331KRLRRVWRRWRMAP-04-0411Cell viability >80% at 50 µM
312023993331KRLRRVWRRWRMAP-04-0411Cell viability >80% at 75 µM
312123993331KRLRRVWRRWRMAP-04-0411Cell viability >80% at 100 µM
312223993331KWLRRVWRWWRMAP-04-0311IC50=61.5 µM
312723770440FLGMIPGLIGGLISAFKTsAP-217IC50 = 6.4 µM
313223770440FLSLIPKLVKKIIKAFKTsAP-S117IC50 = 1.8 µM
313723770440FLGMIPKLIKKLIKAFKTsAP-S217IC50 = 1.8 µM
316023301519WRWRWRWRWCyclic [W(RW)4 ]-Dox960-79% inhibition of cell proliferation at 1 µM
316423301519RWRWRWRWlinear (RW)4-Dox860-74% antiproliferative activity at 1 µM
319117787026(K-Aib-C(CH2CO-2'-Pac))4Dimer of peptide-paclitaxel conjugate3IC50 =0.62nM
319417787026(K-Aib-C(CH2CO-2'-Pac))3Trimer of peptide-paclitaxel conjugate3IC50 =3.00nM
319717787026(K-Aib-C(CH2CO-2'-Pac))4Tetramer of peptide-paclitaxel conjugate3IC50 =0.64nM
321622413859KVKVKVKVpPTKVKVKVKSVS-118IC50 =8.1±0.8 µM
321722413859KVKVKVKVpPTKVKVKVKSVS-118IC50 =5.6±0.5 µM
322022413859kvkvkvkvPptkvkvkvkD-SVS-118IC50 =4.7±0.4 µM
322122413859kvkvkvkvPptkvkvkvkD-SVS-118IC50 =3.2±0.4 µM
322422413859KVKVKVKVPPTKVKVKVKSVS-218IC50 >100 µM
322522413859KVKVKVKVPPTKVKVKVKSVS-218IC50 >100 µM
326918815734VRRFPWWWPFLRRTritrpticin13IC50 =142 µg/ml
327218815734KKKFPWWWPFKKKPST13-RK13IC50 =80 µg/ml
327518815734KKKFPWWWPFKKKCKKKFPWWWPFKKKCdi-PST13-RK-C28IC50 =17 µg/ml
327818815734KKKFPWWWPFKKKKKKFPWWWPFKKKKdi-PST13-RK-K27IC50 =10 µg/ml
330621453492WKKW-Dip-KKWKLTX-3029IC50 =73 ± 2 µM
330921453492KKWWKKW-Dip-KLTX-3159IC50 =31 ± 3 µM
331221453492OOW-Dip-OOWWOLTX-3189IC50 =216 ± 36 µM
331521453492, 23533710FKCRRWQWRMKKLfcinB12IC50 > 160 µM
381622963485MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLAN
NFVLIVSQLQPSQENEMFSIRDSAHRRFLLFRRA
FKQL
wtmda-7/IL-24206Cell viability(% of control)=0.5 at concentration 7 µg/ml
381822963485MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANN
FVLIVSQLQPSQENEMFSIRGDSAHRRFLLFRRAF
KQLDVEAALTKALGEVDILLTWMQKFYKL
RGD-mda-7207Cell viability(% of control)=0.5 at concentration 4 µg/ml
382022963485MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANN
FVLIVSQLQPSQENEMFSIRDSAHRRFLLFRRAF
KQL
wtmda-7/IL-24206Apoptotic rate(%)= >50% at concentration of 8 µg/ml
382322963485MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANNF
VLIVSQLQPSQENEMFSIRGDSAHRRFLLFRRAFK
QLDVEAALTKALGEVDILLTWMQKFYKL
RGD-mda-7207Apoptotic rate(%)= >70% at concentration of 8 µg/ml
387016722632YA*822.4% inhibition at 10-5
387116722632YA*827.5% inhibition at 10-4
389416722632YSA*931.1% inhibition at 10-5
389516722632YSA*931.2% inhibition at 10-4
389616722632YSA*9317.8% inhibition at 10-3
391516722632YSA*1037.7% inhibition at 10-4M
391616722632YSA*10318.7% inhibition at 10-3M
394116722632YSA*G15421.2% inhibition at 10-3M
396516722632YRA*G16415.6% inhibition at 10-3M
399016722632YA*GFM17522.8% inhibition at 10-3M
401516722632YA*GFM1859.6% inhibition at 10-4M
401616722632YA*GFM18529.9% inhibition at 10-3M
402616722632YGGFMA*2362.2% inhibition at 10-6M
402716722632YGGFMA*2367.1% inhibition at 10-5M
402816722632YGGFMA*2366.9% inhibition at 10-4M
402916722632YGGFMA*23625.9% inhibition at 10-3M
403812631273, 9266696GLFDVIKKVASVIGGLCitropin 1.116IC50= 5 M
404712631273, 9266696glfdvikkvasvigglCitropin 1.1D16IC50= 5 M
405612631273, 9266696GLFAVIKKVASVIGGL316IC50= 6 M
406512631273, 9266696GLFDVIKAVASVIGGL516IC50= 5 M
407412631273, 9266696GLFDVIKKVAAVIGGL716IC50= 5 M
408312631273, 9266696GLFDVIKKVASVIKGL1116IC50= 5 M
409212631273, 9266696GLFDVIKKVASVIKKL1316IC50= 5 M
410112631273, 9266696GLFDVIAKVASVIKKL1416IC50= 5 M
411012631273, 9266696GLFAVIKKVASVIKGL1516IC50= 5 M
411912631273, 9266696GLFAVIKKVASVIKKL1616IC50= 5 M
412812631273, 9266696GLFAVIKKVAAVIKKL1716IC50= 5 M
413712631273, 9266696GLFAVIKKVAAVIRRL1816IC50= 5 M
414612631273, 9266696GLFAVIKKVAKVIKKL1916IC50= 5 M
415512631273, 9266696GLFKVIKKVASVIGGL2216IC50= 5 M
416412631273, 9266696GLFKVIKKVAKVIKKL2316IC50= 5 M
417312631273, 9266696LGGIVSAVKKIVDFLGretro16IC50= >10 µM
4336NoneYHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKKEB-Lytic32IC50= 6.5 µM
4342NoneYRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKKEB(H2R)-lytic32IC50= 1.9 µM
4349NoneNYQWVPYQGRVPYPRGGLLkLLKklLKKLlKLSema3A(aa363-377) -nLytic32IC50= 13.1 µM
4353NoneGRVPYPRGGLLkLLKklLKKLlKLSema3A(aa371-377) -nLytic24IC50= 14.1 µM
448522057278KAAKKWAKAAKKWAKAWKKAAZ121EC50 =186 µM
448622057278KAAKKWAKAWKKAAKAWKKAAZ221EC50 =173 µM
448722057278KAAKKAWKAWKKAAKAAWKKAAZ321EC50 =128 µM
448822057278KAAKKAWKAAKKAAKWWKKAAZ421EC50 =68 µM
448922057278KAAKKAWKWAKKAAKWAKKAAZ521EC50 =28 µM
449022057278KWWKKAAKAAKKAAKAAKKWAZ621EC50 =16 µM
449122057278KAAKKAWKAAKKAWKAAKKAAZ721EC50 =15 µM
449222057278AWKKWAKAWKWAKAKWWAKAAZ821EC50 =14 µM
449322057278AAWKWAWAKKWAKAKKWAKAAZ921EC50 =16 µM
449422057278AAKKWAKAKWAKAKKWAKAAZ1021EC50 >211 µM
451122023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-03265% cytotoxic at 5 µM
451222023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-03265% cytotoxic at 10 µM
451322023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032630-35% cytotoxic at 25 µM
451422023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032660% cytotoxic at 50 µM
451522023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-03265-10% cytotoxic at 5 µM
451622023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032610% cytotoxic at 10 µM
451722023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032630-35% cytotoxic at 25 µM
451822023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032660% cytotoxic at 50 µM
451922023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032630% cytotoxic at 5 µM
452022023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032650% cytotoxic at 10 µM
452122023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032670% cytotoxic at 25 µM
452222023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032680-85% cytotoxic at 50 µM
452322023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032630% cytotoxic at 5 µM
452422023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032640-50% cytotoxic at 10 µM
452522023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032660-70% cytotoxic at 25 µM
452622023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032680-85% cytotoxic at 50 µM
452722023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032615-20% cytotoxic at 5 µM
452822023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032640-50% cytotoxic at 10 µM
452922023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032680% cytotoxic at 25 µM
453022023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032685-90% cytotoxic at 50 µM
453122023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-0725~0% cytotoxic at 5 µM
453222023734RWGKWFKKATHVGKHVGKAALTAYLNRC-07255% cytotoxic at 10 µM
453322023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072520-30% cytotoxic at 25 µM
453422023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072540-50% cytotoxic at 50 µM
453522023734RWGKWFKKATHVGKHVGKAALTAYLNRC-0725~0% cytotoxic at 5 µM
453622023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072510% cytotoxic at 10 µM
453722023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072520% cytotoxic at 25 µM
453822023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072540-50% cytotoxic at 50 µM
453922023734RWGKWFKKATHVGKHVGKAALTAYLNRC-0725~0% cytotoxic at 5 µM
454022023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072520% cytotoxic at 10 µM
454122023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072570-80% cytotoxic at 25 µM
454222023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072580-85% cytotoxic at 50 µM
454322023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072510% cytotoxic at 5 µM
454422023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072550% cytotoxic at 10 µM
454522023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072580% cytotoxic at 25 µM
454622023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072580-90% cytotoxic at 50 µM
454722023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072530-40% cytotoxic at 5 µM
454822023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072560-70% cytotoxic at 10 µM
454922023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072580-90% cytotoxic at 25 µM
455022023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072585-90% cytotoxic at 50 µM
455122023734GWRTLLKKAEVKTVGKLALKHYLNRC-1323~5% cytotoxic at 10 µM
455222023734GWRTLLKKAEVKTVGKLALKHYLNRC-132310% cytotoxic at 25 µM
455322023734GWRTLLKKAEVKTVGKLALKHYLNRC-132310-15% cytotoxic at 50 µM
455422023734GWRTLLKKAEVKTVGKLALKHYLNRC-1323~0% cytotoxic at 5 µM
455522023734GWRTLLKKAEVKTVGKLALKHYLNRC-1323~0% cytotoxic at 10 µM
455622023734GWRTLLKKAEVKTVGKLALKHYLNRC-132310% cytotoxic at 25 µM
455722023734GWRTLLKKAEVKTVGKLALKHYLNRC-132310-15% cytotoxic at 50 µM
455822023734GWRTLLKKAEVKTVGKLALKHYLNRC-132310% cytotoxic at 5 µM
455922023734GWRTLLKKAEVKTVGKLALKHYLNRC-132310% cytotoxic at 10 µM
456022023734GWRTLLKKAEVKTVGKLALKHYLNRC-132310-15% cytotoxic at 25 µM
456122023734GWRTLLKKAEVKTVGKLALKHYLNRC-132315-20% cytotoxic at 50 µM
456222023734GWRTLLKKAEVKTVGKLALKHYLNRC-1323~5% cytotoxic at 5 µM
456322023734GWRTLLKKAEVKTVGKLALKHYLNRC-1323~5% cytotoxic at 10 µM
456422023734GWRTLLKKAEVKTVGKLALKHYLNRC-13235% cytotoxic at 25 µM
456522023734GWRTLLKKAEVKTVGKLALKHYLNRC-132310-15% cytotoxic at 50 µM
456622023734GWRTLLKKAEVKTVGKLALKHYLNRC-1323~0% cytotoxic at 5 µM
456722023734GWRTLLKKAEVKTVGKLALKHYLNRC-1323~0% cytotoxic at 10 µM
456822023734GWRTLLKKAEVKTVGKLALKHYLNRC-13235-10% cytotoxic at 25 µM
456922023734GWRTLLKKAEVKTVGKLALKHYLNRC-132320% cytotoxic at 50 µM
457022023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032670% cytotoxic at 50 µM
457122023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072570% cytotoxic at 50 µM
457222023734GWRTLLKKAEVKTVGKLALKHYLNRC-13230% cytotoxic at 50 µM
457322023734GRRKRKWLRRIGKGVKIIGGAALDHLNRC-032660-70% cytotoxic at 50 µM
457422023734RWGKWFKKATHVGKHVGKAALTAYLNRC-072560-70% cytotoxic at 50 µM
457522023734GWRTLLKKAEVKTVGKLALKHYLNRC-1323~5% cytotoxic at 50 µM
459921351323YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKKEGFR-lytic32IC50 =0.12 µM
460021351323YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKKEGFR-lytic32IC50 =0.46 µM
461220802991CSSRTMHHCPeptide-209at 100 µM 55% viablity
461920964334KWKWKWDex-(KW)36at 10 µM 35-40% viablity
467222885172GLFGKLIKKFGRKAISYAVKKARGKHLatarcin 2a26graph fig 8 A
500124587350GIGKFLKKAKKFGKAFVKILKKPexiganan22LC50= 8 at 100 µM
500224587350LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTESLL 3737LC50= 21 at 100 µM
505824830845ETFSDWWKLLAEmt_L22 W/P27A12IC50=16.3 µM
505924830845LTFSDWWKLLAEmt_E17L/L22 W/P27A12IC50=15.1 µM
506024830845ESFSDWWKLLAEmt_T18S/L22 W/P27A12IC50=27 µM
506124830845ETFADWWKLLAEmt_S20A/L22 W/P27A12IC50= 8.7 µM