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IDPMIDSEQUENCENAME LENGTHACTIVITY
110318617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=11.2 µg/ml
110418617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=14.6 µg/ml
110518617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=13.2 µg/ml
110618617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=17.6 µg/ml
110718617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=12 µg/ml
110818617323RAGLQFPVGRLLRRLLRRLLRBuforin IIb21IC50=12.7 µg/ml
12337849420KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKALCecropin B35IC50=25.5 µM
12347849420KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKALCecropin B35IC50=>100 µM
12377849420SWLSKTAKKLENSAKKRISEGIAIAIQGGPRCecropin P131IC50=>100 µM
12387849420SWLSKTAKKLENSAKKRISEGIAIAIQGGPRCecropin P131IC50=>100 µM
12417849420MPRWRLFRRIDRVGKQIKQGILRAGPAIALVGDARAVGShiva-138IC50=49.3 µM
12427849420MPRWRLFRRIDRVGKQIKQGILRAGPAIALVGDARAVGShiva-138IC50=>100 µM
12457849420KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKALCecropin B35IC50=33.5 µM
12477849420KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKALCecropin B35IC50=37 µM
12497849420KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKALCecropin B35IC50=>100 µM
125510951191GLFDIIKKIAESFAurein1.213LC50 = 10 µM
126410951191GLFDIVKKVVGAFGSLAurein2.516LC50=10-100 µM
127310951191GLFDIAKKVIGVIGSLAurein2.616LC50=10-100 µM
128210951191GLFDIVKKIAGHIAGSIAurein 3.117LC50 = 10 µM
129110951191GLFDIVKKIAGHIASSIAurein 3.217LC50=10-100 µM
130010951191GLFDIVKKIAGHIVSSIAurein 3.317LC50 = 10 µM
142816269280KILRGVCKKIMRTFLRRISKDILTGKKNK-227LD50=1-4 µM
147521252288KWKSFAKTFKSAKKTVAHTALKAISSL6A/L17A26IC50=>83.6 µMo/L
147621252288KWKSFLKTFKSAKKTVAHTAAKAISSL17A/L21A26IC50=>83.6 µMo/L
147721252288KWKSFLKTFKSAKKTVAHTALKAISSL17A26IC50=>83.6 µMo/L
147821252288KWKSFLKTFKSAKKTVAHTAAKAISSL21A26IC50=>83.6 µMo/L
147921252288KWKSFAKTFKSAKKTVLHTALKAISSL6A26IC50=>83.6 µMo/L
148021252288KWKSFLKTFKSAKKTVLHTALKAISSP26IC50=11.1 µMo/L
148121252288KWKSFLKTFKSLKKTVLHTALKAISSA12L26IC50=6.4 µMo/L
148221252288KWKSFLKTFKSAKKTVLHTLLKAISSA20L26IC50=5 µMo/L
148321252288KWKSFLKTFKSLKKTVLHTLLKAISSA12L/A20L26IC50=4.3 µMo/L
148421252288KWKSFLKTFKSLKKTVLHTLLKLISSA12L/A20L/A23L26IC50=3.5 µMo/L
154718656352KAQIRAMECNILA512Not Available
154818656352RKKRRQRRRTat9~10% Cytotoxicity at 100 µM
154918656352KAQIRAMECNILGRKKRRQRRRTat-a522~80% Cytotoxicity at 100 µM
163412366526PEWFKCRRWQWRMKKLGAL118IC50=>404 µM
163512366526PAWFKARRWAWRMKKLAAL218IC50=>440 µM
163612366526PAWRKAFRWAWRMKKLAAL318IC50=141 µM
163712366526PAWFKARRWAWRMLKKAAL418IC50=57 µM
163812366526PAWRKAFRWAWRMLKKAAL518IC50=14 µM
163912366526PAWRKAFRWAARMLKKAAL618IC50=15 µM
164012366526PAWRKAFRAAWRMLKKAAL718IC50=16 µM
164112366526PAWAKAFRAAARMKLKAAL818IC50=180 µM
164212366526PAWRKAARWAWRMLKKAAL918IC50=52 µM
164312366526PAARKAFRWAWRMLKKAAL1018IC50=35 µM
164412366526PAARKAARWAWRMLKKGAL1118IC50=248 µM
164512366526PAWRKAFRWAKRMLKKAAL1218IC50=25 µM
164612366526PAWRKAFRKAWRMLKKAAL1318IC50=29 µM
164712366526PAWRKARRWAWRMKKLAAL1418IC50=423 µM
164812366526PAWRKARRWARRMKKLAAL1518IC50=178 µM
166915796184LRVRLASHLRKLRKRLLRDADDLQKRLAVYApo E3065 % Cytotoxity at 40 µg/ml
167022641352LLRHVVKILEKYLTemporin-La1357.62 Inhibition ratio at 50 µg/ml
167122641352LLRHVVKILSKYLTemporin-Las1362.73 Inhibition ratio at 50 µg/ml
167222641352RGDLLRHVVKILEKYLRGD-La1672.69 Inhibition ratio at 50 µg/ml
167322641352RGDLLRHVVKILSKYLRGD-Las1681.465 Inhibition ratio at 50 µg/ml
1734NoneFLGWLFKWAKKGaegurin peptides SEQID NO: 111IC50 = 27 mM
1735NoneFLKWLFKWAKKGaegurin peptides SEQID NO: 211IC50 = 14.8 mM
1736NoneFLGWLFKWAWKGaegurin peptides SEQID NO: 311IC50 = 24.63 mM
1737NoneFLWWLFKWAWKGaegurin peptides SEQID NO: 411IC50 = 14.8 mM
1738NoneFLGWLFKWAKKGaegurin peptides SEQID NO: 111Not Available
1739NoneFLKWLFKWAKKGaegurin peptides SEQID NO: 211Not Available
1740NoneFLGWLFKWAWKGaegurin peptides SEQID NO: 311IC50 = 48 mM
1741NoneFLWWLFKWAWKGaegurin peptides SEQID NO: 411IC50 = 57 mM
1745NoneFLGWLFKWAKKGaegurin peptides SEQID NO: 111Not Available
1751NoneFLKWLFKWAKKGaegurin peptides SEQID NO: 211IC50 = 14.8 mM
1753NoneFLKWLFKWAKKGaegurin peptides SEQID NO: 211Not Available
1759NoneFLGWLFKWAWKGaegurin peptides SEQID NO: 311IC50 = 24.63 mM
1761NoneFLGWLFKWAWKGaegurin peptides SEQID NO: 311IC50 = 48 mM
1767NoneFLWWLFKWAWKGaegurin peptides SEQID NO: 411IC50 = 14.8 mM
1769NoneFLWWLFKWAWKGaegurin peptides SEQID NO: 411IC50 = 57 mM
1925NoneFALALKALKKALKKLKKALKKALHecate AC23LD50 =6 µg/ml
1926NoneFALALKALKKALKKLKKALKKALHecate AM23LD50 =46 µg/ml
1927NoneMPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALGSB-37 AC38LD50 =82 µg/ml
1928NoneMPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALGSB-37 AM38LD50 =>1000 µg/ml
1929NoneFAKKLAKKLKKLAKKLAKLALALSHIVA 10 AC23Not Available
1930NoneFALAAKALKKLAKKLKKLAKKALFLAK01 AM23LD50 =5 µg/ml
1931NoneFALALKALKKLLKKLKKLAKKALFLAK03 AM23LD50 =38 µg/ml
1932NoneFALALKALKKLAKKLKKLAKKALFLAK04 AM23LD50 =12 µg/ml
1933NoneFALAKLAKKAKAKLKKALKALFLAK05 AM21LD50 =8 µg/ml
1934NoneFALALKALKKLKKALKKALFLAK06 AM19LD50 =26 µg/ml
1935NoneFALALKALKKLKKALKKALFLAK06 AC19LD50 =59 µg/ml
1936NoneFAKKLAKKLKKLAKLALALFLAK06 R-AC19LD50 =210 µg/ml
1937NoneVALALKALKKALKKLKKALKKALKAL V23LD50 =62 µg/ml
1938NoneFALALKKALKALKKALFLAK 17 AM16LD50 =35 µg/ml
1939NoneFAKKLAKLAKKLAKLALFLAK 26 AM17LD50 =14 µg/ml
1940NoneFAKKLAKLAKKLAKLALALFLAK 25 AM19LD50 =30 µg/ml
1941NoneFALALKALKKALkkLKKALKKALHECATE 2DAc23LD50 =57 µg/ml
1942NoneFAKKLAKLAKKLLALFLAK43 AM15LD50 =13 µg/ml
1943NoneFAKKLAKLAKKALALFLAK44 AM15LD50 =435 µg/ml
1944NoneFALAKKALKKAKKALFLAK62 AM15LD50 =>1000 µg/ml
1945NoneFAKKLAKKLKKLAKLALAKFLAK 06R-AM19LD50 =120 µg/ml
1946NoneGIGKFLKKAKKFGKAFVKILKKMSI-78 AM22LD50 =34 µg/ml
1947NoneFAKLLAKLAKKLLFLAK5013LD50 =9 µg/ml
1948NoneFAKKLAKLALKLAKLFLAK5115LD50 =32 µg/ml
1949NoneFAKKLAKKLAKLALFLAK5714LD50 =180 µg/ml
1950NoneFAKKLKKLAKLAKKLFLAK7115LD50 =160 µg/ml
1951NoneFAKKALKALKKLFLAK7712LD50 =>1000 µg/ml
1952NoneVAKLLAKLAKKLLFLAK50V13LD50 =47 µg/ml
1953NoneFAKLLAKLAKKLFLAK50F12LD50 =100 µg/ml
1954NoneVAKKLAKLAKKLAKLALFLAK26V AM17LD50 =46 µg/ml
1955NoneKWKLFKKIGAVLKVLCAME-1515Not Available
1956NoneFAKLLAKLAKKALFLAK50C13Not Available
1957NoneFAKLLAKALKKLLFLAK50D13LD50 =14 µg/ml
1958NoneFAKLLKLAAKKLLFLAK 50E13LD50 =215 µg/ml
1959NoneFAKLLAKKLLFLAK8010LD50 =740 µg/ml
1960NoneFAKKLAKALLFLAK8110LD50 =>1000 µg/ml
1961NoneFAKKLAKKLLFLAK8210LD50 =42 µg/ml
1962NoneFAKLAKKLLFLAK83M9LD50 =>1000 µg/ml
1963NoneFAKKLAKLAKKLAKLALFLAK 26 Ac17LD50 =100 µg/ml
1964NoneILPWKWPWWPWRRIndolicidin13LD50 =345 µg/ml
1965NoneFAKALKALLKALKALFLAK 17 C15LD50 = µg/ml
1966NoneFAKLLAKLAKAKLFLAK 50H13LD50 =345 µg/ml
1967NoneFAKLLAKLAKLKLFLAK 50G13LD50 =145 µg/ml
1968NoneFAKKLAKKLKKLAKKLAKKWKLSHIVA DERIV P69 + KWKL22LD50 =11 µg/ml
1969NoneFAKKLAKKLKKLAKKLAKShiva 10(1-18 AC)18LD50 =250 µg/ml
1970NoneFAKKLAKKLKKLAKKLAKKWKLSHIVA 10 PEPTIDE 71 + KWKL22LD50 =82 µg/ml
1971NoneKWKLFKKKTKLFKKFAKKLAKKLCA(1-7) Shiva10(1-16)23LD50 =70 µg/ml
1972NoneFAKKLAKKLAKALFLAK 5413LD50 =340 µg/ml
1973NoneFAKKLAKKLAKLLFLAK 5613LD50 =17 µg/ml
1974NoneFAKKLAKKLAKAALFLAK 5814LD50 =400 µg/ml
1975NoneFAKKLAKKAKLAKKLFLAK 7215LD50 =>1000 µg/ml
1976NoneFAKKLKKLAKKLFLAK 7512LD50 =>1000 µg/ml
1977NoneKTKLFKKFAKKLAKKLKKLAKKLSHIVA 10 (1-16) Ac23LD50 =35 µg/ml
1978NoneKWKLFKKKTKLFKKFAKKLAKKLCA(1-7) Shiva10(1-16)-COOH23LD50 =13 µg/ml
1979NoneILPWKWPWWPWRRIndolocidin-ac13LD50 =30 µg/ml
1980NoneFAKALAKLAKKLLFLAK50B13LD50 =51 µg/ml
1981NoneFAKLLALALKLKLFLAK50I13Not Available
1982NoneFAKLLAKLAKAKAFLAK50K13LD50 =>1000 µg/ml
1983NoneFAKLLAKLAKAKGFLAK50L13LD50 =>1000 µg/ml
1984NoneFAKKLAKKLKKLAKKLAKLALALKALALKALShiva-1131LD50 =125 µg/ml
1985NoneFAKKLAKKLKKLAKKLIGAVLKVSHIVA 11[(1-16)ME(2-9]-COOH23LD50 =120 µg/ml
1986NoneFAKLLAKALKLKLFLAK 50N13LD50 =170 µg/ml
1987NoneFAKLLAKALKKALFLAK 50O13LD50 =57 µg/ml
1988NoneFAKLLAKALKKLFLAK 50P12LD50 =90 µg/ml
1989NoneKWKLFKKALKKLKKALKKALCA(1-& HECATE(11/23)20LD50 =54 µg/ml
1990NoneKIAKVALAKLGIGAVLKVLTTGLPYL-ME23LD50 =>1000 µg/ml
1991NoneFAKKLAKLAKKLFLAG26-D112LD50 =570 µg/ml
1992NoneMPKEKVFLKIEKMGRNIRNVISHNU319LD50 =>1000 µg/ml
1993NoneGIGAVLKVLTTGLPALISWIKRKRQQMELITTIIN26LD50 =23 µg/ml
1994NoneFAKKLAKLAKKLAKALFLAK26-D216LD50 =>1000 µg/ml
1995NoneFAKKLLAKALKLFLAG26-D312LD50 =325 µg/ml
1996NoneFAKFLAKFLKKALFLAK50 Q113LD50 =27 µg/ml
1997NoneFAKLLFKALKKALFLAK50 Q213LD50 =800 µg/ml
1998NoneFAKLLAKFLKKALFLAK50 Q313LD50 =180 µg/ml
1999NoneFAKLLAKAFKKALFLAK50 Q413LD50 =>1000 µg/ml
2000NoneFAKLFAKAFKKALFLAK50 Q513LD50 =>1000 µg/ml
2001NoneFAKLLAKALKKFLFLAK50 Q613LD50 =115 µg/ml
2002NoneFAKLLAKALKKFALFLAK50 Q714LD50 =46 µg/ml
2003NoneFAKLLAKLAKKFALFLAK50 Q814LD50 =630 µg/ml
2004NoneFAKLFAKLAKKFALFLAK50 Q914LD50 =800 µg/ml
2005NoneFKLAFKLAKKAFLFLAK50 Q1013LD50 =570 µg/ml
2006NoneFAKLLAKLAKFLAK50 T110LD50 =>1000 µg/ml
2007NoneFAKLLAKLAKKVLFLAK50 T213LD50 =9 µg/ml
2008NoneFAKLLAKLAKKILFLAK50 T313LD50 =125 µg/ml
2009NoneFAKLLAKLAKKELFLAK50 T413LD50 =>1000 µg/ml
2010NoneFAKLLAKLAKKSLFLAK50 T513LD50 =400 µg/ml
2011NoneFAKLAFLAK905LD50 =530 µg/ml
2012NoneFAKLFFLAK915LD50 =550 µg/ml
2013NoneKAKLFFLAK925LD50 =>1000 µg/ml
2014NoneKWKLFFLAK935LD50 =555 µg/ml
2015NoneFGKGIGKVGKKLLFLAK50 Z113LD50 =>1000 µg/ml
2016NoneFAFGKGIGKVGKKLLFLAK50 Z215LD50 =>1000 µg/ml
2017NoneFAKAIAKIAFGKGIGKVGKKLLFLAK50 Z322LD50 =740 µg/ml
2018NoneFAKLWAKLAFGKGIGKVGKKLLFLAK50 Z422LD50 =80 µg/ml
2019NoneFAKLWAKLAKKLFLAK50 Z512LD50 =600 µg/ml
2020NoneFAKGVGKVGKKALFLAK50 Z613LD50 =>1000 µg/ml
2021NoneFAFGKGIGKIGKKGLFLAK50 Z715LD50 =>1000 µg/ml
2022NoneFAKIIAKIAKIAKKILFLAK50 Z816LD50 =>1000 µg/ml
2023NoneFAFAKIIAKIAKKIIFLAK50 Z915LD50 =>1000 µg/ml
2024NoneFALALKAFLAK947LD50 =560 µg/ml
2025NoneKWKLAKKALALLFLAK93B12LD50 =38 µg/ml
2026NoneFAKIIAKIAKKIFLAK50 Z1012LD50 =>1000 µg/ml
2027NoneFALALKALKKALFLAK9612LD50 =285 µg/ml
2028NoneFALKALKKFLAK978LD50 =>1000 µg/ml
2029NoneKYKKALKKLAKLLFLAK9813LD50 =380 µg/ml
2030NoneFKRLAKIKVLRLAKIKRFKRLA17LD50 =185 µg/ml
2031NoneFAKLAKKALAKLLFLAK91B13LD50 =>1000 µg/ml
2032NoneKAKLAKKALAKLLFLAK92B13LD50 =>1000 µg/ml
2033NoneKLALKLALKALKAAKLAFLAK9917LD50 =235 µg/ml
2034NoneFAKLLAKLAKKFLAK50T611LD50 =>1000 µg/ml
2035NoneFAKLLAKLAKKGLFLAK50T713LD50 =740 µg/ml
2036NoneFALKALKKLKKALKKALFLAK9517LD50 =61 µg/ml
2037NoneVAKLLAKLAKKVLFLAK50T813LD50 =750 µg/ml
2038NoneYAKLLAKLAKKALFLAK50T913LD50 =>1000 µg/ml
2039NoneKLLKLLLKLYKKLLKLLFLAK100-CO2H17LD50 =345 µg/ml
2040NoneFAVGLRAIKRALKKLRRGVRKVAKDLFAGVL26LD50 =530 µg/ml
2041NoneKLAKKLAKLAKLAKALModelin-516LD50 =140 µg/ml
2042NoneKLAKKLAKLAKLAKALModelin-5-CO2H16LD50 =370 µg/ml
2043NoneKWKKLAKKWFLAK1209LD50 =240 µg/ml
2044NoneFALAKALKKALFLAK12111LD50 =>1000 µg/ml
2045NoneFALALKLAKKALFLAK96B12LD50 =360 µg/ml
2046NoneFALLKLFLAK96G6LD50 =>1000 µg/ml
2047NoneFALALKALKKFLAK96F10LD50 =>1000 µg/ml
2048NoneFALKALKKALFLAK96C10LD50 =>1000 µg/ml
2049NoneFALLKALKKALFLAK96D11LD50 =770 µg/ml
2050NoneKFKKLAKKFModelin-8D9LD50 =>1000 µg/ml
2051NoneKFKKLAKKWModelin-8E9LD50 =70 µg/ml
2052NoneFALALKALKKAFlak 96H11LD50 =>1000 µg/ml
2053NoneFALLKALLKKALFlak 96I12LD50 =310 µg/ml
2054NoneFALALKLAKKLFlak 96J11LD50 =>1000 µg/ml
2055NoneLKKLAKLALAFFlak 96L11LD50 =>1000 µg/ml
2056NoneVALALKALKKLFLAK-120G11LD50 =600 µg/ml
2057NoneFALALKLKKLFLAK-120D10LD50 =870 µg/ml
2058NoneFALALKAKKLFLAK-120C10LD50 =>1000 µg/ml
2059NoneFALAFLAK-120B4LD50 =>1000 µg/ml
2060NoneWALALFLAK-120F5LD50 =440 µg/ml
2061NoneGIGKFLHAAKKFAKAFVAEIMNSMagainin2wisc23LD50 =60 µg/ml
2062NoneFAKKFAKKFKKFAKKFAKFAFAFD2A2123LD50 =76 µg/ml
2063NoneKKVVFKVKFKKSL-110LD50 =>1000 µg/ml
2064NoneFKVKFKVKVKKSL-710LD50 =530 µg/ml
2065NoneLPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALGLSB-3738LD50 =240 µg/ml
2066NoneFAKKLAKKLKKLAKKLAKLAKKLAnubis-223LD50 =73 µg/ml
2067NoneFAKKLAKLAKKLAKLALALFLAK 17 CV19Not Available
2068NoneVAKFLAKFLKKALFLAK50 Q1V13Not Available
2069NoneVAKKFAKKFKKFAKKFAKFAFAFD2A21V23Not Available
2070NoneFAKKLAKLAKKLAKLALALFLAK 25 AM V19Not Available
2071NoneFAKKLAKLAKKLLALFLAK43 AM V15Not Available
2072NoneVAKLLAKALKKLLFLAK50D V13Not Available
2073NoneVALALKALKKALKKLKKALKKALHecate AM V23Not Available
2074NoneVALALKALKKALKKLKKALKKALHecate AC V23Not Available
2075NoneFALALKALKKLAKKLKKLAKKALFLAK04 AM V23Not Available
2076NoneFAKLLAKLAKKAAFLAK50J13Not Available
310222783018PDEDAINNALNKVCSTGRRQRSICKQLLKKN29N30100% cell viability at 5 µM
310322783018PDEDAINNALNKVCSTGRRQRSICKQLLKKN29N3040% cell viability at 50 µM
310822783018PDEDAINDALNKVCSTGRRQRSICKQLLKKN29D30>100% cell viability at 5 µM
310922783018PDEDAINDALNKVCSTGRRQRSICKQLLKKN29D3060% cell viability at 50 µM
315923301519WRWRWRWRWCyclic [W(RW)4 ]-Dox950-67% inhibition of cell proliferation at 1 µM
316323301519RWRWRWRWlinear (RW)4-Dox821-61% antiproliferative activity at 1 µM
317517559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 54016.5 % inhibition of cell proliferation at 1 nM
317617559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 54014.2 % inhibition of cell proliferation at 10 nM
317717559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 54016.8 % inhibition of cell proliferation at 100 nM
317817559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 54021.7 % inhibition of cell proliferation at 1 µM
317917559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 54027.9 % inhibition of cell proliferation at 10 µM
318717559067fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HLPeptide 540ED50 >10 µM
322822644847FLGWLFKWAWKGA-W311IC50 =24.63 µM
323522644847FLWWLFKWAWKGA-W411IC50 =14.80 µM
324222644847FLGWLFKWAKKGA-K311IC50 =27.00 µM
324922644847FLKWLFKWAKKGA-K411IC50 =14.80 µM
325422783018PDEDAINNALNKVCSTGRRQRSICKQLLKKN29N30100% cell viability at 5 µM
325522783018PDEDAINNALNKVCSTGRRQRSICKQLLKKN29N3040% cell viability at 50 µM
326022783018PDEDAINDALNKVCSTGRRQRSICKQLLKKN29D30>100% cell viability at 5 µM
326122783018PDEDAINDALNKVCSTGRRQRSICKQLLKKN29D3060% cell viability at 50 µM
328119527490, 23533710FKCRRWQWRMKKLfcinB12IC50 =148±8 µM
328919527490KAAKKAAKAAKKAAKAAKKAAKW521IC50 =55±14 µM
330521453492WKKW-Dip-KKWKLTX-3029IC50 =75 ± 5 µM
330821453492KKWWKKW-Dip-KLTX-3159IC50 =38 ± 3 µM
331121453492OOW-Dip-OOWWOLTX-3189IC50 =248 ± 5 µM
331421453492, 23533710FKCRRWQWRMKKLfcinB12IC50 > 160 µM
334123533710FKCRRWQWRMKKLfcinB12Inhibition at 0.1g/l
334223533710YPFPGβ-Casomorphins 5 f(60_64)4Inhibition at 9-11g/l
334323533710RYLGYLαs1-casein f(90_95)6Inhibition at 12-15g/l
334423533710PPPEECaseinphosphopeptides5Inhibition at 24-28g/l
3362NoneNHFTLKCPKTALTEPPTLAYTG2020<5% cytotoxicity at 1 µM
3363NoneNHFTLKCPKTALTEPPTLAYTG2020<20% cytotoxicity at 10 µM
3364NoneNHFTLKCPKTALTEPPTLAYTG2020~15% cytotoxicity at 1 µM
3365NoneNHFTLKCPKTALTEPPTLAYTG2020>20% cytotoxicity at 10 µM
3366NoneNHFTLKCPKTALTEPPTLAYTG2020<5% cytotoxicity at 1 µM
3367NoneNHFTLKCPKTALTEPPTLAYTG2020<5% cytotoxicity at 10 µM
3368NoneTAGIKLTVPIEKFPVTTQTFWGTG2322<5% cytotoxicity at 1 µM
3369NoneTAGIKLTVPIEKFPVTTQTFWGTG2322~10% cytotoxicity at 10 µM
3370NoneTAGIKLTVPIEKFPVTTQTFWGTG232210% cytotoxicity at 1 µM
3371NoneTAGIKLTVPIEKFPVTTQTFWGTG2322>10% cytotoxicity at 10 µM
3372NoneTAGIKLTVPIEKFPVTTQTFWGTG2322>10% cytotoxicity at 1 µM
3373NoneTAGIKLTVPIEKFPVTTQTFWGTG2322<5% cytotoxicity at 10 µM
3374NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030<5% cytotoxicity at 1 µM
3375NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030<5% cytotoxicity at 10 µM
3376NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030>20% cytotoxicity at 1 µM
3377NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030~35% cytotoxicity at 10 µM
3378NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030<5% cytotoxicity at 1 µM
3379NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030~20% cytotoxicity at 10 µM
3398NoneNHFTLKCPKTALTEPPTLAYTG202020% cytotoxicity at 1 µM
3399NoneNHFTLKCPKTALTEPPTLAYTG202010% cytotoxicity at 10 µM
3400NoneNHFTLKCPKTALTEPPTLAYTG2020<5% cytotoxicity at 1 µM
3401NoneNHFTLKCPKTALTEPPTLAYTG2020<3% cytotoxicity at 10 µM
3402NoneNHFTLKCPKTALTEPPTLAYTG2020<20% cytotoxicity at 1 µM
3403NoneNHFTLKCPKTALTEPPTLAYTG202015% cytotoxicity at 10 µM
3404NoneTAGIKLTVPIEKFPVTTQTFWGTG2322<15% cytotoxicity at 1 µM
3405NoneTAGIKLTVPIEKFPVTTQTFWGTG232215% cytotoxicity at 10 µM
3406NoneTAGIKLTVPIEKFPVTTQTFWGTG2322~5% cytotoxicity at 1 µM
3407NoneTAGIKLTVPIEKFPVTTQTFWGTG2322<5% cytotoxicity at 10 µM
3408NoneTAGIKLTVPIEKFPVTTQTFWGTG2322<5% cytotoxicity at 1 µM
3409NoneTAGIKLTVPIEKFPVTTQTFWGTG2322<5% cytotoxicity at 10 µM
3410NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030>40% cytotoxicity at 1 µM
3411NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB303050% cytotoxicity at 10 µM
3412NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030<20% cytotoxicity at 1 µM
3413NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030>20% cytotoxicity at 10 µM
3414NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030>30% cytotoxicity at 1 µM
3415NoneGQVWEATATVNAIRGSVTPAVSQFNARTADMB3030~40% cytotoxicity at 10 µM
351922100226VNWKKILGKIIKVVKLL-III/3715IC50 = 5±1 µM
352022100226VNWKKILGKIIKVVKLL-III15IC50 = 18±4 µM
352122100226VNWKKILAKIIKVVKLL-III/115IC50 = 12± 3 µM
352222100226NVWKKILGKIIKVVKLL-III/215IC50 = 11 µM
352322100226VNWKKILKKIIKVVKLL-III/315IC50 > 40 µM
352422100226VNWKKILGKIKKVVKLL-III/415IC50 > 40 µM
352522100226VNWKKILPKIIKVVKLL-III/615Not tested
352622100226VNWKKILGKIIKVVKLL-III/815Not tested
352722100226VNWKKILGKIIKVVKLL-III/915IC50 = 25± 5 µM
352822100226KNWKKILGKIIKVVKLL-III/1015Not tested
352922100226VNWKKIILGKIIKVVKLL-III/1115IC50 = 48 µM
353022100226vnwkkilgkiikvvkLL-III/1215IC50 = 20 µM
353122100226VNFKKLLGKLLKVVKLL-III/1515IC50 = 42 µM
353222100226VN-Nal-KKLLGKLLKVVKLL-III/1615Not tested
353322100226VNWRRILGRIIRVVRLL-III/1715Not tested
353422100226KNWKKILKKIIKVVKLL-III/1815Not tested
353522100226VNWKK-Aib-LGK-Aib-IK-Aib-VKLL-III/1915IC50 = 28 µM
353622100226KNWKK-Aib-LKK-Aib-IK-Aib-VKLL-III/2215IC50 > 100 µM
353722100226VNWKKLLGKLLKVVKLL-III/2315IC50 = 15 µM
353822100226VNWOOILGOIIOVVOLL-III/2415IC50 = 20 µM
353922100226vnwkkllgkllkvvkLL-III/2515IC50 = 20 µM
354022100226VYWKKILGKIIKVVKLL-III/2615IC50 = 30 µM
354122100226VNWKKVLGKVVKVVKLL-III/2715IC50 > 100 µM
354222100226NKWKKILGKIIKVVKLL-III/3415IC50 = 37 µM
354322100226VNWKKILAKIIKVVKLL-III/3615Not tested
354422100226VNWKKILGKIIKVVKLL-III/3715IC50 = 13 µM
360222100226GFGMALKLLKKVLMAC113IC50 = 23±4 µM
360322100226GTGLPMSERRKIMLMMRMAC217IC50 > 100 µM
360422100226gfgmalkllkkvlMAC1/113IC50 = 19±2 µM
360522100226AFGMALKLLKKVLMAC1/213IC50 = 16 µM
360622100226LFGMALKLLKKVLMAC1/313IC50 = 11±1 µM
360722100226GFGMALKLLKKVLMAC1/413IC50 = 49±9 µM
360822100226GFGMALKLLKKVLMAC1/613IC50 = 29±3 µM
360922100226GFKMALKLLKKVLMAC1/913IC50 = 13±3 µM
361022100226GFKMALKLLKKVLMAC1/1013Not tested
361122100226GFGMALKLLKKVLMAC1/1613IC50 > 100 µM
361222100226GFGMALKLLKKVLMAC1/1913IC50 = 68±2 µM
361322100226GFGMALOLLOOVLMAC1/2013IC50 = 35±4 µM
361422100226GFGMALRLLRRVLMAC1/2113IC50 = 17±2 µM
361522100226GFGMALKL-(AC6C)-KKVLMAC1/2413IC50 = 16±1 µM
361622100226GFGMALK-(AC6C)-LKKVLMAC1/2513IC50 = 14±1 µM
361722100226GFGMA-(AC6C)-KLLKKVLMAC1/2613IC50 = 18±1 µM
366222100226GMWSKILGHLIRHAL-112IC50 = 44±8 µM
366322100226gmwskilghlirHAL-1/2212IC50 > 40 µM
366422100226GMWSKILGHLIKHAL-1/612IC50 > 100 µM
366522100226GMWSKILGHLKRHAL-1/412Not tested
366622100226GMWSKILGKLIRHAL-1/912IC50 > 50 µM
366722100226GMWSKILKHLIRHAL-1/1812IC50 = 18±2 µM
366822100226GMWKKILGHLIRHAL-1/512IC50 = 44±5 µM
366922100226GKWSKILGHLIRHAL-1/1212IC50 > 100 µM
367022100226KMWSKILGHLIRHAL-1/1712IC50 > 100 µM
367122100226GMWKKILGKLIRHAL-1/1012IC50 > 60 µM
367222100226GKWSKILGKLIRHAL-1/2012IC50 > 40 µM
367322100226GKWKKILGHLIRHAL-1/1912IC50 > 100 µM
367422100226GKWKKILGKLIRHAL-1/2112IC50 > 100 µM
367522100226GMWSKILGHLIRHAL-1/2912Not tested
367622100226GMWSKLLGHLLRHAL-1/1512IC50 > 40 µM
367722100226GKWMSLLKHILKHAL-212IC50 = 35±3 µM
367822100226gkwmsllkhilkHAL-2/2212IC50 > 100 µM
367922100226GKWMSLLKKILKHAL-2/412IC50 = 38±6 µM
368022100226GKWMKLLKHILKHAL-2/212IC50 = 35±5 µM
368122100226GKWKSLLKHILKHAL-2/112IC50 > 100 µM
368222100226GKWMSLLKHILKHAL-2/812IC50 > 40 µM
368322100226GKWMSLLKHIWKHAL-2/1812IC50 > 40 µM
368422100226GKWMSLLKHWLKHAL-2/1912IC50 > 40 µM
368522100226GKWMSLWKHILKHAL-2/2012IC50 > 40 µM
368622100226GKFMSLLKHILKHAL-2/2412IC50 > 40 µM
368722100226GKWMSFLKHILKHAL-2/612IC50 > 40 µM
368822100226GKWMTLLKHILKHAL-2/1312IC50 > 60 µM
368922100226GKWLSLLKHILKHAL-2/1112IC50 = 40 µM
37249815815fA*YwKA*TLan-77IC50= 29.97±1.19 µM
372922644847FLGWLFKWAWKGA-W311IC50= 24.63 µM
373622644847FLWWLFKWAWKGA-W411IC50= 14.80 µM
374322644847FLGWLFKWAKKGA-K311IC50= 27.00 µM
375022644847FLKWLFKWAKKGA-K411IC50= 14.8 µM
385816722632YA*829.8% inhibition at 10-6
385916722632YA*821.6% inhibition at 10-5
386016722632YA*825.4% inhibition at 10-4
386116722632YA*8226.5% inhibition at 10-3
386216722632YA*8212.9% inhibition at 10-6
386316722632YA*8216.5% inhibition at 10-5
386416722632YA*8228.1% inhibition at 10-4
386516722632YA*8258.2% inhibition at 10-3
386616722632YA*823.5% inhibition at 10-6
386716722632YA*8222.7% inhibition at 10-5
386816722632YA*8218.9% inhibition at 10-4
386916722632YA*8226.4% inhibition at 10-3
388216722632YSA*934.9% inhibition at 10-6
388316722632YSA*938.9% inhibition at 10-5
388416722632YSA*933.4% inhibition at 10-4
388516722632YSA*9320.8% inhibition at 10-3
388616722632YSA*9310.5% inhibition at 10-6
388716722632YSA*9321.9% inhibition at 10-5
388816722632YSA*9311.8% inhibition at 10-4
388916722632YSA*9317.9% inhibition at 10-3
389016722632YSA*933.7% inhibition at 10-6
389116722632YSA*9316.5% inhibition at 10-5
389216722632YSA*938.4% inhibition at 10-4
389316722632YSA*9314.5% inhibition at 10-3
390916722632YSA*1030.7% inhibition at 10-6
391016722632YSA*1038.3% inhibition at 10-5
391116722632YSA*10310.5% inhibition at 10-4
391216722632YSA*10321.8% inhibition at 10-3
391316722632YSA*10310.7% inhibition at 10-6
391416722632YSA*10310.0% inhibition at 10-5
392916722632YSA*G1545.4% inhibition at 10-6M
393016722632YSA*G1547.4% inhibition at 10-5M
393116722632YSA*G1549.5% inhibition at 10-4M
393216722632YSA*G15415.7% inhibition at 10-3M
393316722632YSA*G15413.6% inhibition at 10-6M
393416722632YSA*G15420.4% inhibition at 10-5M
393516722632YSA*G15414.4% inhibition at 10-4M
393616722632YSA*G15423.4% inhibition at 10-3M
393716722632YSA*G1542.2% inhibition at 10-6M
393816722632YSA*G1544.2% inhibition at 10-5M
393916722632YSA*G1546.4% inhibition at 10-4M
394016722632YSA*G1546.2% inhibition at 10-3M
395316722632YRA*G1647.6% inhibition at 10-6M
395416722632YRA*G1643.8% inhibition at 10-5M
395516722632YRA*G16412.4% inhibition at 10-4M
395616722632YRA*G16422.4% inhibition at 10-3M
395716722632YRA*G16417.0% inhibition at 10-6M
395816722632YRA*G16413.5% inhibition at 10-5M
395916722632YRA*G16413.5% inhibition at 10-4M
396016722632YRA*G16425.3% inhibition at 10-3M
396116722632YRA*G1648.1% inhibition at 10-6M
396216722632YRA*G1646.9% inhibition at 10-5M
396316722632YRA*G1648.1% inhibition at 10-4M
396416722632YRA*G1648.6% inhibition at 10-3M
397816722632YA*GFM1753.3% inhibition at 10-6M
397916722632YA*GFM17511.0% inhibition at 10-5M
398016722632YA*GFM1757.9% inhibition at 10-4M
398116722632YA*GFM17523.7% inhibition at 10-3M
398216722632YA*GFM17512.2% inhibition at 10-6M
398316722632YA*GFM17515.5% inhibition at 10-5M
398416722632YA*GFM17524.7% inhibition at 10-4M
398516722632YA*GFM17529.0% inhibition at 10-3M
398616722632YA*GFM1753.0% inhibition at 10-6M
398716722632YA*GFM1758.4% inhibition at 10-5M
398816722632YA*GFM17518.5% inhibition at 10-4M
398916722632YA*GFM17510.6% inhibition at 10-3M
400316722632YA*GFM18516.2% inhibition at 10-6M
400416722632YA*GFM1856.6% inhibition at 10-5M
400516722632YA*GFM1855.1% inhibition at 10-4M
400616722632YA*GFM18514.5% inhibition at 10-3M
400716722632YA*GFM18526.4% inhibition at 10-6M
400816722632YA*GFM18513.1% inhibition at 10-5M
400916722632YA*GFM18514.6% inhibition at 10-4M
401016722632YA*GFM18538.4% inhibition at 10-3M
401116722632YA*GFM18517.7% inhibition at 10-6M
401216722632YA*GFM18510.9% inhibition at 10-5M
401316722632YA*GFM18512.1% inhibition at 10-4M
401416722632YA*GFM1858.1% inhibition at 10-3M
402316722632YGGFMA*2369.2% inhibition at 10-3M
402416722632YGGFMA*23611.08% inhibition at 10-5M
402516722632YGGFMA*23647.0% inhibition at 10-3M
403212631273, 9266696GLFDVIKKVASVIGGLCitropin 1.116IC50= 5 M
404112631273, 9266696glfdvikkvasvigglCitropin 1.1D16IC50= 5 M
405012631273, 9266696GLFAVIKKVASVIGGL316IC50= 6 M
405912631273, 9266696GLFDVIKAVASVIGGL516IC50= 5 M
406812631273, 9266696GLFDVIKKVAAVIGGL716IC50= 5 M
407712631273, 9266696GLFDVIKKVASVIKGL1116IC50= 5 M
408612631273, 9266696GLFDVIKKVASVIKKL1316IC50= 5 M
409512631273, 9266696GLFDVIAKVASVIKKL1416IC50= 5 M
410412631273, 9266696GLFAVIKKVASVIKGL1516IC50= 5 M
411312631273, 9266696GLFAVIKKVASVIKKL1616IC50= 5 M
412212631273, 9266696GLFAVIKKVAAVIKKL1716IC50= 5 M
413112631273, 9266696GLFAVIKKVAAVIRRL1816IC50= 5 M
414012631273, 9266696GLFAVIKKVAKVIKKL1916IC50= 5 M
414912631273, 9266696GLFKVIKKVASVIGGL2216IC50= 5 M
415812631273, 9266696GLFKVIKKVAKVIKKL2316IC50= 5 M
416712631273, 9266696LGGIVSAVKKIVDFLGretro16IC50= >10 µM
449522057278KAAKKWAKAAKKWAKAWKKAAZ121EC50 >211 µM
449622057278KAAKKWAKAWKKAAKAWKKAAZ221EC50 >211 µM
449722057278KAAKKAWKAWKKAAKAAWKKAAZ321EC50 >211 µM
449822057278KAAKKAWKAAKKAAKWWKKAAZ421EC50 =173 µM
449922057278KAAKKAWKWAKKAAKWAKKAAZ521EC50 =67 µM
450022057278KWWKKAAKAAKKAAKAAKKWAZ621EC50 =31 µM
450122057278KAAKKAWKAAKKAWKAAKKAAZ721EC50 =21 µM
450222057278AWKKWAKAWKWAKAKWWAKAAZ821EC50 =23 µM
450322057278AAWKWAWAKKWAKAKKWAKAAZ921EC50 =13 µM
450422057278AAKKWAKAKWAKAKKWAKAAZ1021EC50 >211 µM
457821423613PRFWEYWLRLMEMIP12IC50 =0.01 µM
457921423613LTFEHYWAQLTSDI12IC50 =0.29 µM
458021423613LTAEHYAAQATS3A12IC50 >100 µM
458121423613QETFSDLWKLLPP5317-2812IC50 =4.7 µM
458221423613PRAWEYWLRLMEMIP(F3A)12IC50 =0.57 µM
458321423613PRFWEAWLRLMEMIP(Y6A)12IC50 >100 µM
458421423613PRFWEYALRLMEMIP(W7A)12IC50 >100 µM
458521423613PRFWEYWLALMEMIP(R9A)12IC50 =0.02 µM
458621423613PRFWEYWLRAMEMIP(L10A)12IC50 =1.14 µM
458721423613PRFWEYWLRLAEMIP(M11A)12IC50 =0.4 µM
458821423613PRFWEYWLRLMEMIP12IC50 =0.12 µM
458921423613LTFEHYWAQLTSDI12IC50 =1.6 µM
459021423613LTAEHYAAQATS3A12IC50 >100 µM
459121423613QETFSDLWKLLPP5317-2812IC50 =30 µM
501624962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >50% at 25μM approx
501724962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability =50% at 12.5μM approx.
501824962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >50% at 12.5μM approx.
501924962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >60% at 25μM approx
502024962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >50% at 25μM approx
502124962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >60% at 25μM approx
502224962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >60% at 25μM approx
502324962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >50% at 25μM approx
502424962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >50% at 25μM approx
502524962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >50% at 25μM approx
502624962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >50% at 25μM approx
502724962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >50% at 25μM approx
502824962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >60% at 25μM approx
502924962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability =50% at 12.5μM approx.
503024962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability =50% at 12.5μM approx.
503124962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >40% at 12.5μM approx
503224962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >40% at 12.5μM approx
503324962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >50% at 12.5μM approx
503424962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >55% at 12.5μM approx
503524962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >55% at 12.5μM approx
503624962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >75% at 12.5μM approx
503724962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >55% at 12.5μM approx
503824962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >55% at 12.5μM approx
503924962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >70% at 12.5μM approx
504024962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >45% at 12.5μM approx
504124962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >80% at 12.5μM approx
504224962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >85% at 12.5μM approx
504324962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >70% at 12.5μM approx
504424962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >60% at 12.5μM approx
504524962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >70% at 12.5μM approx
504624962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >80% at 12.5μM approx
504724962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >65% at 12.5μM approx
504824962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >70% at 12.5μM approx
504924962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >55% at 12.5μM approx
505024962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >80% at 12.5μM approx
505124962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >85% at 12.5μM approx
505224962950KILRGVAKKIMRTFLRRISKDILTGKKC7A27Cell viability >50% at 12.5μM approx
505324962950KILRGVAKKIMRTFLRRISKKILTGKKC7A-D21K27Cell viability >65% at 12.5μM approx
505424962950KILRGVAKKIMRTFLRRISKDILTGKKC7A-Δ27Cell viability >70% at 12.5μM approx
505624714081TKPRKTKPRKTKPRKTKPRT Peptide1970% maximum inhibitory rate at 8 mg/kg