Details of CPPsite entry with Sequence HHHHHHHHHHHHRRRRRRRRRRRRRRR |
| Primary information | |
|---|---|
| PEPTIDE SEQUENCE | HHHHHHHHHHHHRRRRRRRRRRRRRRR |
| CPPsite ID | 2137, |
| PEPTIDE NAME | STR-H12R8 |
| CHIRALITY | L |
| LINEAR/CYCLIC | Linear |
| SOURCE | Synthetic |
| CATEGORY | Cationic |
| SUB CELLULAR LOCALIZATION | Cytoplasm |
| N-TERMINAL MODIFICATION | Stearylation |
| C-TERMINAL MODIFICATION | Amidation |
| UPTAKE EFFICIENCY | STR-H12R8 induced gene silencing with the knockdown efficiency of 31% at R/P 5 and 59% at R/P 10 |
| PROPOSED UPTAKE MECHANISM | Endocytosis |
| INVITRO/INVIVO | In vitro |
| CELL LINE | CHO-K1 cells, HeLa |
| CARGO | Nucleic acid (GAPDH siRNA) |
| PMID | 25193363 |
| PATENT | Unknown |
| Tertiary Structure (Technique) | 2137 (PEPstrMOD), |