Details of CPPsite entry with Sequence PKKKRKV-AGYLLGKINLKALAALAKKIL-PQMQQNVFQYPGAGMVPQGEANF |
| Primary information | |
|---|---|
| PEPTIDE SEQUENCE | PKKKRKV-AGYLLGKINLKALAALAKKIL-PQMQQNVFQYPGAGMVPQGEANF |
| CPPsite ID | 2264, 2266, |
| PEPTIDE NAME | TP10-SRC1LXXLL, TP10-SRC1(1222-1245) |
| CHIRALITY | L, L |
| LINEAR/CYCLIC | Linear, Linear |
| SOURCE | Chimeric, Chimeric |
| CATEGORY | Cationic, Cationic |
| SUB CELLULAR LOCALIZATION | Cytoplasm and Nucleus, Cytoplasm and Nucleus |
| N-TERMINAL MODIFICATION | Conjugated with NLS, Conjugated with NLS |
| C-TERMINAL MODIFICATION | Free, Free |
| CHEMICAL MODIFICATION | NA, NA |
| UPTAKE EFFICIENCY | Higher uptake efficiency, Lower uptake efficiency than TP10-SRC1LXXLL |
| PROPOSED UPTAKE MECHANISM | NA, NA |
| INVITRO/INVIVO | In vitro, In vitro |
| CELL LINE | MCF-7 cells, MCF-7 cells |
| In VIVO MODEL | NA, NA |
| CARGO | Fluorophore (FITC ), Fluorophore (FITC ) |
| PMID | 24705462, 24705462 |
| PATENT | Unknown, Unknown |
| Tertiary Structure (Technique) | 2264 (PEPstrMOD), 2266 (I-TASSER), |