| NO. | Protein Target | Peptide |
| 1. | Atrial natriuretic peptide receptor A | Nesiritide |
| 2. | Atrial natriuretic peptide receptor B | Nesiritide |
| 3. | Atrial natriuretic peptide clearance receptor | Nesiritide |
| 4. | Cholecystokinin type A receptor | Ceruletide |
| 5. | Pancreatic triacylglycerol lipase | Bentiromide |
| 6. | Glucagon-like peptide 1 receptor | Exenatide |
| 7. | Glucagon | Exenatide |
| 8. | Gonadotropin-releasing hormone receptor | Gonadorelin |
| 9. | Gonadotropin-releasing hormone II receptor | Gonadorelin |
| 10. | Envelope glycoprotein | Enfuvirtide |
| 11. | Dihydropyrimidine dehydrogenase [NADP+] | Enfuvirtide |
| 12. | DNA | Vancomycin |
| 13. | Glycosyltransferase GtfA | Vancomycin |
| 14. | Aminopeptidase N | Icatibant |
| 15. | B2 bradykinin receptor | Icatibant |
| 16. | Secretin receptor | Secretin |
| 17. | Gonadotropin-releasing hormone receptor
| Leuprolide |
| 18. | Glucagon receptor | Glucagon recombinant |
| 19. | Glucagon-like peptide 1 receptor | Glucagon recombinant |
| 20. | Carboxypeptidase E | Glucagon recombinant |
| 21. | Glucagon-like peptide 2 receptor | Glucagon recombinant |
| 22. | Oxytocin-neurophysin | Oxytocin |
| 23. | Prolyl endopeptidase | Oxytocin |
| 24. | Prothrombin | Bivalirudin |
| 25. | Growth hormone-releasing hormone receptor
| Sermorelin |
| 26. | 50S ribosomal protein L10 | Capreomycin |
| 27. | Calcitonin receptor | Salmon Calcitonin |
| 28. | Vasopressin V1a receptor | Vasopressin |
| 29. | Vasopressin V2 receptor | Vasopressin |
| 30. | Vasopressin V1b receptor | Vasopressin |
| 31. | Adrenocorticotropic hormone receptor | Cosyntropin |
| 32. | Probable low molecular weight protein-tyrosine-phosphatase epsP | Bacitracin |
| 33. | Alpha-2-macroglobulin | Bacitracin |
| 34. | Protachykinin 1 | Bacitracin |
| 35. | Insulin-degrading enzyme | Bacitracin |
| 36. | Somatostatin receptor type 1 | Octreotide |
| 37. | Somatostatin receptor type 5 | Octreotide |
| 38. | Substance-K receptor | Octreotide |
| 39. | Gonadotropin-releasing hormone receptor | Abarelix |
| 40. | Substance-P receptor | Vapreotide |
| 41. | Lutropin-choriogonadotropic hormone receptor | Cetrorelix |
| 42. | Gonadotropin-releasing hormone receptor | Cetrorelix |
| 43. | Parathyroid hormone/parathyroid hormone-related peptide receptor | Teriparatide |
| 44. | Adrenocorticotropic hormone receptor
| Corticotropin |
| 45. | Lutropin-choriogonadotropic hormone receptor | Goserelin |
| 46. | Vasopressin V1a receptor | Desmopressin |
| 46. | Vasopressin V1b receptor | Desmopressin |
| 47. | Receptor activity-modifying protein 1 | Pramlintide |
| 48. | Receptor activity-modifying protein 2 | Pramlintide |
| 49. | Receptor activity-modifying protein 3 | Pramlintide |
| 50. | Growth hormone receptor | Pegvisomant |
| 51. | Prolactin receptor | Pegvisomant |
| 52. | Growth hormone receptor | Somatropin recombinant |
| 53. | Prolactin receptor | Somatropin recombinant |
| 54. | Lutropin-choriogonadotropic hormone receptor | Lutropin alfa |
| 55. | Follicle-stimulating hormone receptor | Follitropin beta |
| 56. | Follicle-stimulating hormone receptor | Urofollitropin |
| 57. | Lutropin-choriogonadotropic hormone receptor | Menotropins |
| 58. | Follicle-stimulating hormone receptor | Menotropins |
| 59. | Thyrotropin receptor | Thyrotropin Alfa |
| 60. | Lutropin-choriogonadotropic hormone receptor | Choriogonadotropin alfa |
| 61. | Follicle-stimulating hormone receptor | Choriogonadotropin alfa |
| 62. | Interferon-alpha/beta receptor beta chain | Interferon Alfa-2a, Recombinant |
| 63. | Interferon-alpha/beta receptor alpha chain | Interferon Alfa-2a, Recombinant |
| 63. | Interferon-alpha/beta receptor beta chain | Interferon alfacon-1 |
| 64. | Interferon-alpha/beta receptor alpha chain | Interferon alfacon-1 |
| 65. | Interferon-alpha/beta receptor beta chain | Interferon Alfa-2b, Recombinant |
| 66. | Interferon-alpha/beta receptor alpha chain | Interferon Alfa-2b, Recombinant |
| 67. | Interferon-alpha/beta receptor beta chain | Interferon beta-1b |
| 68. | Interferon-alpha/beta receptor alpha chain | Interferon beta-1b |
| 69. | Interferon-alpha/beta receptor beta chain | Interferon alfa-n3 |
| 70. | Interferon-alpha/beta receptor alpha chain | Interferon alfa-n3 |
| 71. | Interferon-alpha/beta receptor beta chain | Interferon alfa-n1 |
| 72. | Interferon-alpha/beta receptor alpha chain | Interferon alfa-n1 |
| 73. | Interferon-gamma receptor beta chain | Interferon alfa-n1 |
| 74. | Interferon-alpha/beta receptor alpha chain | Peginterferon alfa-2b |
| 75. | Interferon-alpha/beta receptor beta chain | Peginterferon alfa-2b |
| 76. | Interferon-alpha/beta receptor alpha chain | Peginterferon alfa-2a |
| 77. | Interferon-alpha/beta receptor beta chain | Peginterferon alfa-2a |
| 78. | Interleukin-2 receptor subunit beta | Aldesleukin |
| 79. | Interleukin-2 receptor alpha chain | Aldesleukin |
| 80. | Cytokine receptor common gamma chain | Aldesleukin |
| 81. | Coagulation factor VIII | Coagulation Factor IX |
| 82. | Prothrombin | Coagulation Factor IX |
| 83. | Coagulation factor X | Coagulation Factor IX |
| 84. | Coagulation factor VII | Coagulation Factor IX |
| 85. | Vitamin K-dependent gamma-carboxylase | Coagulation Factor IX |
| 86. | Coagulation factor XI | Coagulation Factor IX |
| 87. | Low-density lipoprotein receptor-related Protein 1 | Coagulation Factor IX |