ID | PEPTIDE SEQUENCE | PEPTIDE NAME | LENGTH | CHIRALITY | LINEAR/CYCLIC | SOURCE | CATEGORY | N TERMINAL MODIFICATION | C TERMINAL MODIFICATION | CHEMICAL MODIFICATION | CARGO | PUBMED ID |
---|---|---|---|---|---|---|---|---|---|---|---|---|
2009 | WRWKKKKA | cyclic [W(RW)4] | 8 | L | Cyclic | Synthetic | Cationic | NA | NA | Drug conjugated with peptide through linker | Small molecule drug (Doxorubicin) | 23301519 |
2125 | CHHRRRRHHC | CH2 R4 H2 C | 10 | L | Cyclic | Synthetic | NA | Stearylation | Free | NA | Nucleic aciud (siRNA) | 23911914 |
2167 | CSKSSDYQC | CSK | 9 | L | Cyclic | Synthetic | NA | Free | Free | Coupling to polyoxyethylene (40) steartae (SA-PEG2000) | Nanoparticle [salmon calcitonin (sCT)-loaded SLNs (Solid Lipid Nanoparticle)] | 24968819 |
2169 | CGYGRKKRRQRRRGC | TAT | 15 | L | Cyclic | Protein derived | Cationic | Free | Free | NA | Nucleic acid (pDNA) | 24985759 |
2240 | Cyclo (FΦRRRRQ) | cFΦR4-Rho | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine | Fluorophore (Rhodamine), Protein (GFP) | 24896852 |
2241 | Cyclo (FΦRRRRQ) | cFΦR4-Dex | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine | Dexamethasone | 24896852 |
2242 | GRKKRRQRRRPPQY | Tat-Dex | 14 | L | Cyclic | Protein derived | Cationic | Free | Amidation | Dexamethasone | Dexamethasone | 24896852 |
2243 | Cyclo(FΦRRRRQ) | cFΦR4-FITC | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine | Fluorophore (FITC) | 24896852 |
2244 | Cyclo (FΦRRRRQ) | cFΦR4-R5 | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine | Peptide (RRRRR) | 24896852 |
2245 | Cyclo (FΦRRRRQ) | cFΦR4-A5 | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine | Peptide (AAAAA) | 24896852 |
2246 | Cyclo (FΦRRRRQ) | cFΦR4-F4 | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine | Peptide (FFFF) | 24896852 |
2247 | Cyclo (FΦRRRRQ) | cFΦR4-PCP | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine,miniPEG, 8-amino-3,6-dioxaoctanoic acid | Peptide [PCP, miniPEG-DE(pCAP)LI-NH2] | 24896852 |
2251 | Cyclo (FΦRRRRQ) | bicyclo(FΦR4-A5)Rho | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine, J, l-2,3-diaminopropionic acid, Tm, trimesoyl | Cyclic peptide (Tm(AAAAA)) | 24896852 |
2252 | Cyclo (FΦRRRRQ) | bicyclo(FΦR4-A7)Rho | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine, J, l-2,3-diaminopropionic acid, Tm, trimesoyl | Cyclic peptide Tm(AAAAAAA)K | 24896852 |
2253 | Cyclo (FΦRRRRQ) | bicyclo(FΦR4-RARAR)Rho | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine, J, l-2,3-diaminopropionic acid, Tm, trimesoyl | Cyclic peptide Tm(RARAR)K | 24896852 |
2254 | Cyclo (FΦRRRRQ) | bicyclo(FΦR4-DADAD)Rho | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine, J, l-2,3-diaminopropionic acid, Tm, trimesoyl | Cyclic peptide Tm(DADAD)K | 24896852 |
2255 | Cyclo (FΦRRRRQ) | monocyclo(FΦR4-A5)Rho | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine | Peptide AAAAA | 24896852 |
2256 | Cyclo (FΦRRRRQ) | monocyclo(FΦR4-A7)Rho | 8 | Modified | Cyclic | Synthetic | Amphipathic | Free | Amidation | Φ, L-2-naphthylalanine | Peptide AAAAAAA | 24896852 |
2298 | RGDfK | cRGD | 5 | L | Cyclic | Protein derived | NA | Cycliclization | Cyclization | NA | Fluorophore (Alexa488), Protein (bovine serum albumin) and Nanoparticle (quantum dots) | 25108152 |
2349 | ACSGSGSGCGSGSGSCG | IA0 (Bicyclic) (integral arginine peptides) | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2350 | ACSGRGSGCGSGRGSCG | IA2 | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2351 | ACRGSGRGCGRGSGRCG | IA4a | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2352 | ACSGRGRGCGRGRGSCG | IA4b | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2353 | ACRGRGRGCGRGRGRCG | IA6a | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2354 | ACGRGRGRCRGRGRGCG | IA6b | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2355 | ACRGRGRGCRGRGRGCG | IA6c | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2356 | ACGRGRGRCGRGRGRCG | IA6d | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2357 | ACRGRRRGCGRRRGRCG | IA8a | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2358 | ACRRSRRGCGRRSRRCG | IA8b | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2359 | ACSDRFRNCPADEALCG | kCA2 (Kallikrein inhibitor with internal arginines) | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2360 | ACRDRFRNCPADEALCG | kCA3 | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2361 | ACRDRFRNCPADERLCG | kCA4 | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2362 | ACRDRFRRCPADERLCG | kCA5 | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2363 | ACRDRFRRCPADRRLCG | kCA6 | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2364 | ACSGRGRGCGSGSGSCG | CA2 (Control internal arginine ) | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2365 | ACRGRGRGCGSGSGSCG | CA3 | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2366 | ACRGRGRGCGSGSRSCG | CA4 | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2367 | ACRGRGRRCGSGSRSCG | CA5 | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2368 | ACRGRGRRCGSGRRSCG | CA6 | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2369 | ARCSGSGSGCGSGSGSCGR | EA2x1 (External arginines) | 19 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2370 | ARRCSGSGSGCGSGSGSCGRR | EA2x2 | 21 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2371 | ARRRCSGSGSGCGSGSGSCGRRR | EA2x3 | 23 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2372 | ARRRRCSGSGSGCGSGSGSCGRRRR | EA2x4 | 25 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2373 | ACSGSGSGCGSGSGSCGRRRRRRRR | EA1x8 | 25 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2374 | ARCSDRFRNCPADEALCGR | kEA2x1 (Kallikrein inhibitor with external arginines) | 19 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2375 | ARRCSDRFRNCPADEALCGRR | kEA2x2 | 21 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2376 | ARRRCSDRFRNCPADEALCGRRR | kEA2x3 | 23 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2377 | ARRRRCSDRFRNCPADEALCGRRRR | kEA2x4 | 25 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2378 | ACSDRFRNCPADEALCGRRRRRRRR | kEA1 8 | 25 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | NA | Fluorophore (FITC) | 24697151 |
2379 | ACRRSRRGCGRRSRRCG | IA8b L (Linear variants) | 17 | L | Cyclic | Synthetic | Arginine rich | Extended with Alanine and an 6-aminohexanoic acid (Ahx) spacer | Amidation | All cysteines were capped with iodoacetamide | Fluorophore (FITC) | 24697151 |