SMDBid | siRNA (sense/antisense) 5'>3' | Modification (sense/antisense) | Position (sense/antisense) |
Modified component (sense/antisense) |
Efficacy (%) | Reference |
SM3478 |
AACCCACCACAGCUAGAACUU AAGUUCUAGCUGUGGUGGGUU |
2-O-Methyl 0 |
14 0 |
Sugar 0 |
84 percent target mRNA inhibition | US20120088815A1, EP2415869A1 |
SM3481 |
AACCCACCACAGCUAGAACUU AAGUUCUAGCUGUGGUGGGUU |
2-O-Methyl 0 |
14 0 |
Sugar 0 |
82 percent target mRNA inhibition | US20120088815A1, EP2415869A1 |
SM3622 |
GACCACGAAGAGUUAACCCTT GGGUUAACUCUUCGUGGUCTT |
2-Deoxy-2-Fluoro 2-Deoxy-2-Fluoro |
14 5 |
Sugar Sugar |
82 percent target mRNA inhibition | US20120088815A1, EP2415869A1 |
SM3694 |
CCGAGAGCUCUCCUACCUUTT AAGGUAGGAGAGCUCUCGGTT |
2-O-Methyl 2-O-Methyl |
14 5 |
Sugar Sugar |
75 percent target mRNA inhibition | US20120088815A1, EP2415869A1 |
SM3758 |
AGAAAAGCAGCGAUACGCUTT AGCGUAUCGCUGCUUUUCUTT |
2-O-Methyl 0 |
14 0 |
Sugar 0 |
69 percent target mRNA inhibition | US20120088815A1, EP2415869A1 |
SM3805 |
CCUCGGAGAGUUCUACUCUTT AGAGUAGAACUCUCCGAGGTT |
2-O-Methyl 2-O-Methyl |
14 5 |
Sugar Sugar |
85 percent target mRNA inhibition | US20120088815A1, EP2415869A1 |
SM3862 |
AUCGUCGUCAGGGUAAGGUTT ACCUUACCCUGACGACGAUTT |
2-O-Methyl 2-O-Methyl |
14 5 |
Sugar Sugar |
49 percent target mRNA inhibition | US20120088815A1, EP2415869A1 |
SM3870 |
GACAAGGGAAGGUUAGCCUTT AGGCUAACCUUCCCUUGUCTT |
2-O-Methyl 2-O-Methyl |
14 5 |
Sugar Sugar |
72 percent target mRNA inhibition | US20120088815A1, EP2415869A1 |
SM3970 |
AGAGAGGUGGAGGUAUCUCTT GAGAUACCUCCACCUCUCUTT |
2-O-Methyl 2-O-Methyl |
14 5 |
Sugar Sugar |
90 percent target mRNA inhibition | US20120088815A1, EP2415869A1 |
SM4218 |
CCGAAGACGAAGCUAUGAATT UUCAUAGCUUCGUCUUCGGTT |
2-O-Methyl 2-O-Methyl |
14 3 |
Sugar Sugar |
71 percent target mRNA inhibition | US20120088815A1, EP2415869A1 |